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21 . Periodical
Bioreductive prodrug PR-104 improves the tumour distribution and titre of the nitroreductase-armed oncolytic adenovirus ONYX-411NTRleading to therapeutic benefit
저자
by
Singleton, Dean C.
;
Mowday, Alexandra M.
;
Guise, Chris P.
;
Syddall, Sophie P.
;
Bai, Sally Y.
, et al.
소스
Cancer Gene Therapy; July 2022, Vol. 29 Issue: 7 p1021-1032, 12p
Web of Science
Scopus
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27 . Academic Journal
Tissue Pharmacokinetic Properties and Bystander Potential of Hypoxia-Activated Prodrug CP-506 by Agent-Based Modelling.
저자
by
Jackson-Patel, Victoria
;
Liu, Emily
;
Bull, Matthew R.
;
Ashoorzadeh, Amir
;
Bogle, Gib
, et al.
소스
Frontiers in Pharmacology; 2/8/2022, Vol. 13, p1-17, 17p
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27 . Academic Journal
Discovery of Cysteine-targeting Covalent Protein Kinase Inhibitors.
저자
by
Xiaoyun Lu
;
Smaill, Jeff B.
;
Patterson, Adam V.
;
Ke Ding
.
소스
Journal of Medicinal Chemistry; 1/13/2022, Vol. 65 Issue 1, p58-83, 26p
Full Text (ACS)
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26 . Academic Journal
Use of an optimised enzyme/prodrug combination for Clostridia directed enzyme prodrug therapy induces a significant growth delay in necrotic tumours
저자
by
Mowday, Alexandra M.
;
Dubois, Ludwig J.
;
Kubiak, Aleksandra M.
;
Chan-Hyams, Jasmine V. E.
;
Guise, Christopher P.
, et al.
소스
Cancer Gene Therapy
. 29(2):178-188
Web of Science
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27 . Academic Journal
Allosterische Kinaseinhibitoren – Erwartungen und Chancen.
저자
by
Lu, Xiaoyun
;
Smaill, Jeff B.
;
Ding, Ke
.
소스
Angewandte Chemie
. 8/10/2020, Vol. 132 Issue 33, p13868-13881. 14p.
Full Text (Wiley)
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25 . Academic Journal
New Promise and Opportunities for Allosteric Kinase Inhibitors.
저자
by
Lu, Xiaoyun
;
Smaill, Jeff B.
;
Ding, Ke
.
소스
Angewandte Chemie International Edition
. 8/10/2020, Vol. 59 Issue 33, p13764-13776. 13p.
Full Text (Wiley)
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25 . Academic Journal
Synthesis and structure–activity relationships of soluble 8-substituted 4-(2-chlorophenyl)-9-hydroxypyrrolo[3,4- c]carbazole-1,3(2 H,6 H)-diones as inhibitors of the Wee1 and Chk1 checkpoint kinases
저자
by
Smaill, Jeff B.
;
Lee, Ho H.
;
Palmer, Brian D.
;
Thompson, Andrew M.
;
Squire, Christopher J.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2008 18(3):929-933
Full Text (ScienceDirect)
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27 . Academic Journal
Directed evolution of the B. subtilis nitroreductase YfkO improves activation of the PET-capable probe SN33623 and CB1954 prodrug.
저자
by
Rich, Michelle H.
;
Sharrock, Abigail V.
;
Ashoorzadeh, Amir
;
Patterson, Adam V.
;
Smaill, Jeff B.
, et al.
소스
Biotechnology Letters; 2021, Vol. 43 Issue 1, p203-211, 9p
Web of Science
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27 . Academic Journal
Small-Molecule Inhibitors Directly Targeting KRAS as Anticancer Therapeutics.
저자
by
Chen, Hao
;
Smaill, Jeff B.
;
Liu, Tongzheng
;
Ding, Ke
;
Lu, Xiaoyun
.
소스
Journal of Medicinal Chemistry; 12/10/2020, Vol. 63 Issue 23, p14404-14424, 21p
Full Text (ACS)
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27 . Academic Journal
The synthesis and biological evaluation of novel series of nitrile-containing fluoroquinolones as antibacterial agents
저자
by
Murphy, Sean T.
;
Case, Heather L.
;
Ellsworth, Edmund
;
Hagen, Susan
;
Huband, Michael
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2007 17(8):2150-2155
Full Text (ScienceDirect)
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