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1 . Academic Journal
Cell-based assays for kinase drug discovery
저자
by
Smith, Gary K.
;
Wood, Edgar R.
.
소스
In
Drug Discovery Today: Technologies
2010 7(1):e13-e19
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4 . Academic Journal
A Scintillation Proximity Assay for the Raf/MEK/ERK Kinase Cascade: High-Throughput Screening and Identification of Selective Enzyme Inhibitors
저자
by
McDonald, Octerloney B.
;
Chen, Wen Ji
;
Ellis, Byron
;
Hoffman, Christine
;
Overton, Laurie
, et al.
소스
In
Analytical Biochemistry
15 March 1999 268(2):318-329
Full Text (ScienceDirect)
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7 . Academic Journal
2,3,5-Trisubstituted pyridines as selective AKT inhibitors—Part I: Substitution at 2-position of the core pyridine for ROCK1 selectivity
저자
by
Lin, Hong
;
Yamashita, Dennis S.
;
Zeng, Jin
;
Xie, Ren
;
Wang, Wenyong
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2010 20(2):673-678
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7 . Academic Journal
Synthesis and evaluation of aniline headgroups for alkynyl thienopyrimidine dual EGFR/ErbB-2 kinase inhibitors
저자
by
Waterson, Alex G.
;
Petrov, Kimberly G.
;
Hornberger, Keith R.
;
Hubbard, Robert D.
;
Sammond, Douglas M.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2009 19(5):1332-1336
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7 . Academic Journal
Thienopyrimidine-based dual EGFR/ErbB-2 inhibitors
저자
by
Rheault, Tara R.
;
Caferro, Thomas R.
;
Dickerson, Scott H.
;
Donaldson, Kelly H.
;
Gaul, Michael D.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2009 19(3):817-820
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7 . Academic Journal
Synthesis and stereochemical effects of pyrrolidinyl-acetylenic thieno[3,2- d]pyrimidines as EGFR and ErbB-2 inhibitors
저자
by
Stevens, Kirk L.
;
Alligood, Krystal J.
;
Alberti, Jennifer G. Badiang
;
Caferro, Thomas R.
;
Chamberlain, Stanley D.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2009 19(1):21-26
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7 . Academic Journal
Dual EGFR/ErbB-2 inhibitors from novel pyrrolidinyl-acetylenic thieno[3,2- d]pyrimidines
저자
by
Hubbard, Robert D.
;
Dickerson, Scott H.
;
Emerson, Holly K.
;
Griffin, Robert J.
;
Reno, Michael J.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2008 18(21):5738-5740
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7 . Academic Journal
Optimization and SAR for dual ErbB-1/ErbB-2 tyrosine kinase inhibition in the 6-furanylquinazoline series
저자
by
Petrov, Kimberly G.
;
Zhang, Yue-Mei
;
Carter, Malcolm
;
Cockerill, G. Stuart
;
Dickerson, Scott
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2006 16(17):4686-4691
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7 . Academic Journal
Alkynyl pyrimidines as dual EGFR/ErbB2 kinase inhibitors
저자
by
Waterson, Alex G.
;
Stevens, Kirk L.
;
Reno, Michael J.
;
Zhang, Yue-Mei
;
Boros, Eric E.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2006 16(9):2419-2422
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7 . Academic Journal
Discovery and in vitro evaluation of potent kinase inhibitors: Pyrido[1′,2′:1,5]pyrazolo[3,4- d]pyrimidines
저자
by
Alberti, Michael J.
;
Auten, Elizabeth P.
;
Lackey, Karen E.
;
McDonald, Octerloney B.
;
Wood, Edgar R.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2005 15(16):3778-3781
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