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1 . Academic Journal
Structure-based optimization of indoline-containing compounds as second generation inhibitors of NF-κB-inducing kinase (NIK)
저자
by
Cheng, Jing
;
Yan, Ziqin
;
Li, Xinzhi
;
Liu, Chen
;
Tong, Linjiang
, et al.
소스
In
Journal of Molecular Structure
5 January 2024 1295 Part 1
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7 . Academic Journal
Preclinical and early clinical studies of a novel compound SYHA1813 that efficiently crosses the blood–brain barrier and exhibits potent activity against glioblastoma
저자
by
Liu, Yingqiang
;
Zhan, Zhengsheng
;
Kang, Zhuang
;
Li, Mengyuan
;
Lv, Yongcong
, et al.
소스
In
Acta Pharmaceutica Sinica B
December 2023 13(12):4748-4764
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7 . Academic Journal
Design and synthesis of 1H-pyrazolo[3,4-d]pyrimidine derivatives as hematopoietic progenitor kinase 1 (HPK1) inhibitors
저자
by
Zhang, Junjie
;
Li, Yan
;
Tang, Haotian
;
Zhou, Qianqian
;
Tong, Linjiang
, et al.
소스
In
Bioorganic Chemistry
November 2023 140
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7 . Academic Journal
Application of deep generative model for design of Pyrrolo[2,3-d] pyrimidine derivatives as new selective TANK binding kinase 1 (TBK1) inhibitors
저자
by
Song, Shukai
;
Tang, Haotian
;
Ran, Ting
;
Fang, Feng
;
Tong, Linjiang
, et al.
소스
In
European Journal of Medicinal Chemistry
5 February 2023 247
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7 . Academic Journal
Discovery of N-(3-bromo-1H-indol-5-yl)-quinazolin-4-amine as an effective molecular skeleton to develop reversible/irreversible pan-HER inhibitors
저자
by
Tang, Qidong
;
Peng, Ting
;
Hu, Jie
;
Zhang, Tao
;
Chen, Pengqin
, et al.
소스
In
European Journal of Medicinal Chemistry
5 April 2022 233
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7 . Academic Journal
Design and synthesis of selective degraders of EGFRL858R/T790M mutant
저자
by
Zhang, Xin
;
Xu, Fang
;
Tong, Linjiang
;
Zhang, Tao
;
Xie, Hua
, et al.
소스
In
European Journal of Medicinal Chemistry
15 April 2020 192
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7 . Academic Journal
Pyrazolo[4,3-b]pyrimido[4,5-e][1,4]diazepine derivatives as new multi-targeted inhibitors of Aurora A/B and KDR
저자
by
Zhang, Qiumeng
;
Shen, Qianqian
;
Gao, Lixin
;
Tong, Linjiang
;
Li, Jia
, et al.
소스
In
European Journal of Medicinal Chemistry
5 October 2018 158:428-441
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7 . Academic Journal
Discovery of novel 2,4-diarylaminopyrimidine derivatives as potent and selective epidermal growth factor receptor (EGFR) inhibitors against L858R/T790M resistance mutation
저자
by
Yan, Qi
;
Chen, Yuzhe
;
Tang, Baiyou
;
Xiao, Qiang
;
Qu, Rong
, et al.
소스
In
European Journal of Medicinal Chemistry
25 May 2018 152:298-306
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7 . Academic Journal
Structure-based design and synthesis of 2,4-diaminopyrimidines as EGFR L858R/T790M selective inhibitors for NSCLC
저자
by
Chen, Lingfeng
;
Fu, Weitao
;
Feng, Chen
;
Qu, Rong
;
Tong, Linjiang
, et al.
소스
In
European Journal of Medicinal Chemistry
10 November 2017 140:510-527
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7 . Academic Journal
A structure-guided optimization of pyrido[2,3-d]pyrimidin-7-ones as selective inhibitors of EGFRL858R/T790M mutant with improved pharmacokinetic properties
저자
by
Yu, Lei
;
Huang, Minhao
;
Xu, Tianfeng
;
Tong, Linjiang
;
Yan, Xiao-e
, et al.
소스
In
European Journal of Medicinal Chemistry
27 January 2017 126:1107-1117
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