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1 . Academic Journal
Synthesis and structure-activity relationships for a new class of tetrahydronaphthalene amide inhibitors of Mycobacterium tuberculosis
저자
by
Sutherland, Hamish S.
;
Lu, Guo-Liang
;
Tong, Amy S.T.
;
Conole, Daniel
;
Franzblau, Scott G.
, et al.
소스
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European Journal of Medicinal Chemistry
5 February 2022 229
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7 . Academic Journal
Structure-activity relationships for analogs of the tuberculosis drug bedaquiline with the naphthalene unit replaced by bicyclic heterocycles
저자
by
Sutherland, Hamish S.
;
Tong, Amy S.T.
;
Choi, Peter J.
;
Conole, Daniel
;
Blaser, Adrian
, et al.
소스
In
Bioorganic & Medicinal Chemistry
1 May 2018 26(8):1797-1809
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7 . Academic Journal
Synthesis and evaluation of analogues of the tuberculosis drug bedaquiline containing heterocyclic B-ring units
저자
by
Choi, Peter J.
;
Sutherland, Hamish S.
;
Tong, Amy S.T.
;
Blaser, Adrian
;
Franzblau, Scott G.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 December 2017 27(23):5190-5196
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7 . Academic Journal
3,5-Dialkoxypyridine analogues of bedaquiline are potent antituberculosis agents with minimal inhibition of the hERG channel.
저자
by
Sutherland, Hamish S.
;
Tong, Amy S.T.
;
Choi, Peter J.
;
Blaser, Adrian
;
Conole, Daniel
, et al.
소스
Bioorganic & Medicinal Chemistry
. Apr2019, Vol. 27 Issue 7, p1292-1307. 16p.
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7 . Academic Journal
Structure-activity relationships for unit C pyridyl analogues of the tuberculosis drug bedaquiline.
저자
by
Blaser, Adrian
;
Sutherland, Hamish S.
;
Tong, Amy S.T.
;
Choi, Peter J.
;
Conole, Daniel
, et al.
소스
Bioorganic & Medicinal Chemistry
. Apr2019, Vol. 27 Issue 7, p1283-1291. 9p.
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7 . Academic Journal
Synthesis and structure-activity relationships for tetrahydroisoquinoline-based inhibitors of Mycobacterium tuberculosis.
저자
by
Lu, Guo-Liang
;
Tong, Amy S.T.
;
Conole, Daniel
;
Sutherland, Hamish S.
;
Choi, Peter J.
, et al.
소스
Bioorganic & Medicinal Chemistry
. Nov2020, Vol. 28 Issue 22, pN.PAG-N.PAG. 1p.
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7 . Academic Journal
Synthetic Studies to Help Elucidate the Metabolism of the Preclinical Candidate TBAJ-876—A Less Toxic and More Potent Analogue of Bedaquiline.
저자
by
Choi, Peter J.
;
Conole, Daniel
;
Sutherland, Hamish S.
;
Blaser, Adrian
;
Tong, Amy S.T.
, et al.
소스
Molecules
. 3/15/2020, Vol. 25 Issue 6, p1423. 1p.
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7 . Academic Journal
Variations in the C-unit of bedaquiline provides analogues with improved biology and pharmacology.
저자
by
Sutherland, Hamish S.
;
Tong, Amy S.T.
;
Choi, Peter J.
;
Blaser, Adrian
;
Franzblau, Scott G.
, et al.
소스
Bioorganic & Medicinal Chemistry
. Jan2020, Vol. 28 Issue 1, pN.PAG-N.PAG. 1p.
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