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1 . Academic Journal
Interactions of hydrolyzed β-lactams with the L1 metallo-β-lactamase: Crystallography supports stereoselective binding of cephem/carbapenem products
저자
by
Hinchliffe, Philip
;
Calvopiña, Karina
;
Rabe, Patrick
;
Mojica, Maria F.
;
Schofield, Christopher J.
, et al.
소스
In
Journal of Biological Chemistry
May 2023 299(5)
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7 . Academic Journal
In silico design of novel quinazoline-based compounds as potential Mycobacterium tuberculosis PknB inhibitors through 2D and 3D-QSAR, molecular dynamics simulations combined with pharmacokinetic predictions
저자
by
Hanwarinroj, Chayanin
;
Thongdee, Paptawan
;
Sukchit, Darunee
;
Taveepanich, Somjintana
;
Kamsri, Pharit
, et al.
소스
In
Journal of Molecular Graphics and Modelling
September 2022 115
Full Text (ScienceDirect)
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7 . Academic Journal
Faropenem reacts with serine and metallo-β-lactamases to give multiple products
저자
by
Lucic, Anka
;
Hinchliffe, Philip
;
Malla, Tika R.
;
Tooke, Catherine L.
;
Brem, Jürgen
, et al.
소스
In
European Journal of Medicinal Chemistry
5 April 2021 215
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7 . Academic Journal
Electric Fields Are a Key Determinant of Carbapenemase Activity in Class A β‑Lactamases.
저자
by
Jabeen, Hira
;
Beer, Michael
;
Spencer, James
;
van der Kamp, Marc W.
;
Bunzel, H. Adrian
, et al.
소스
ACS Catalysis; 5/3/2024, Vol. 14 Issue 9, p7166-7172, 7p
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7 . Academic Journal
Rational Design of Benzobisheterocycle Metallo-β-Lactamase Inhibitors: A Tricyclic Scaffold Enhances Potency against Target Enzymes.
저자
by
Villamil, Valentina
;
Rossi, Maria-Agustina
;
Mojica, Maria F.
;
Hinchliffe, Philip
;
Martínez, Verónica
, et al.
소스
Journal of Medicinal Chemistry; 3/14/2024, Vol. 67 Issue 5, p3795-3812, 18p
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7 . Report
Ab-initio quantum chemistry with neural-network wavefunctions
저자
by
Hermann, Jan
;
Spencer, James
;
Choo, Kenny
;
Mezzacapo, Antonio
;
Foulkes, W. M. C.
, et al.
소스
Open Access (Arxiv)
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7 . Academic Journal
Working together: why language policies of international schools must evolve to incorporate collaborative strategies between EAL and the mainstream.
저자
by
Spencer, James
.
소스
Journal of Research in International Education; Dec2023, Vol. 22 Issue 3, p222-239, 18p
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3 . Academic Journal
Preclinical evaluation of the SARS-CoV-2 M
pro
inhibitor RAY1216 shows improved pharmacokinetics compared with nirmatrelvir
저자
by
Chen, Xiaoxin
;
Huang, Xiaodong
;
Ma, Qinhai
;
Kuzmič, Petr
;
Zhou, Biao
, et al.
소스
Nature Microbiology
. 9(4):1075-1088
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7 . Periodical
Imitation of β-lactam binding enables broad-spectrum metallo-β-lactamase inhibitors
저자
by
Brem, Jürgen
;
Panduwawala, Tharindi
;
Hansen, Jon Ulf
;
Hewitt, Joanne
;
Liepins, Edgars
, et al.
소스
Nature Chemistry; 20240101, Issue: Preprints p1-10, 10p
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7 . Academic Journal
Enhancement by pyrazolones of colistin efficacy against mcr-1-expressing E. coli: an in silico and in vitro investigation.
저자
by
Hanpaibool, Chonnikan
;
Ounjai, Puey
;
Yotphan, Sirilata
;
Mulholland, Adrian J.
;
Spencer, James
, et al.
소스
Journal of Computer-Aided Molecular Design
. Oct2023, Vol. 37 Issue 10, p479-489. 11p.
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