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1 . Academic Journal
Antimalarial activity of single-dose DSM265, a novel plasmodium dihydroorotate dehydrogenase inhibitor, in patients with uncomplicated Plasmodium falciparum or Plasmodium vivax malaria infection: a proof-of-concept, open-label, phase 2a study
저자
by
Llanos-Cuentas, Alejandro
;
Casapia, Martin
;
Chuquiyauri, Raúl
;
Hinojosa, Juan-Carlos
;
Kerr, Nicola
, et al.
소스
In
The Lancet Infectious Diseases
August 2018 18(8):874-883
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7 . Academic Journal
DSM265 for Plasmodium falciparum chemoprophylaxis: a randomised, double blinded, phase 1 trial with controlled human malaria infection
저자
by
Sulyok, Mihály
;
Rückle, Thomas
;
Roth, Alexandra
;
Mürbeth, Raymund E
;
Chalon, Stephan
, et al.
소스
In
The Lancet Infectious Diseases
June 2017 17(6):636-644
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7 . Academic Journal
Safety, tolerability, pharmacokinetics, and activity of the novel long-acting antimalarial DSM265: a two-part first-in-human phase 1a/1b randomised study
저자
by
McCarthy, James S
;
Lotharius, Julie
;
Rückle, Thomas
;
Chalon, Stephan
;
Phillips, Margaret A
, et al.
소스
In
The Lancet Infectious Diseases
June 2017 17(6):626-635
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7 . Academic Journal
Inactivation of PI3Kγ and PI3Kδ distorts T-cell development and causes multiple organ inflammation
저자
by
Ji, Hong
;
Rintelen, Felix
;
Waltzinger, Caroline
;
Bertschy Meier, Dominique
;
Bilancio, Antonio
, et al.
소스
In
Blood
15 October 2007 110(8):2940-2947
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7 . Academic Journal
Key role of the p110δ isoform of PI3K in B-cell antigen and IL-4 receptor signaling: comparative analysis of genetic and pharmacologic interference with p110δ function in B cells
저자
by
Bilancio, Antonio
;
Okkenhaug, Klaus
;
Camps, Montserrat
;
Emery, Juliet L.
;
Ruckle, Thomas
, et al.
소스
In
Blood
15 January 2006 107(2):642-650
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7 . Academic Journal
Sequential activation of class IB and class IA PI3K is important for the primed respiratory burst of human but not murine neutrophils
저자
by
Condliffe, Alison M.
;
Davidson, Keith
;
Anderson, Karen E.
;
Ellson, Chris D.
;
Crabbe, Tom
, et al.
소스
In
Blood
15 August 2005 106(4):1432-1440
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7 . Academic Journal
Synthesis and characterization of constrained cyclosporin A derivatives containing a pseudo-proline group
저자
by
Patiny, Luc
;
Guichou, Jean-François
;
Keller, Michael
;
Turpin, Olivier
;
Rückle, Thomas
, et al.
소스
In
Tetrahedron
2003 59(28):5241-5249
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7 . Academic Journal
Efficacy and safety of temelimab in multiple sclerosis: Results of a randomized phase 2b and extension study.
저자
by
Hartung, Hans-Peter
;
Derfuss, Tobias
;
Cree, Bruce AC
;
Sormani, Maria Pia
;
Selmaj, Krzysztof
, et al.
소스
Multiple Sclerosis Journal
. Mar2022, Vol. 28 Issue 3, p429-440. 12p.
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7 . Academic Journal
Pseudo-prolines in cyclic peptides: Conformational stabilisation of cyclo[Pro-Thr(ψ Me,Mepro)-Pro]
저자
by
Rückle, Thomas
;
de Lavallaz, Pierre
;
Keller, Michael
;
Dumy, Pascal
;
Mutter, Manfred
.
소스
In
Tetrahedron
1999 55(37):11281-11288
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7 . Academic Journal
PI3Kgamma (PI3Kγ) is essential for efficient induction of CXCR3 on activated T cells
저자
by
Barbi, Joseph
;
Cummings, Hannah E.
;
Lu, Bao
;
Oghumu, Steve
;
Rückle, Thomas
, et al.
소스
In
Blood
15 October 2008 112(8):3048-3051
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