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1 . Academic Journal
Characterisation of cotadutide's dual GLP‐1/glucagon receptor agonistic effects on glycaemic control using an in vivo human glucose regulation quantitative systems pharmacology model.
저자
by
Bosch, Rolien
;
Petrone, Marcella
;
Arends, Rosalin
;
Vicini, Paolo
;
Sijbrands, Eric J. G.
, et al.
소스
British Journal of Pharmacology
. Feb2024, p1. 12p. 5 Illustrations, 3 Charts.
Full Text (Wiley)
Web of Science
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7 . Academic Journal
Durable responses to ATR inhibition with ceralasertib in tumors with genomic defects and high inflammation.
저자
by
Dillon, Magnus T.
;
Guevara, Jeane
;
Mohammed, Kabir
;
Patin, Emmanuel C.
;
Smith, Simon A.
, et al.
소스
Journal of Clinical Investigation
. 1/16/2024, Vol. 134 Issue 2, p1-14. 14p.
Web of Science
Scopus
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7 . Academic Journal
Pharmacokinetics and Safety of Cotadutide, a GLP-1 and Glucagon Receptor Dual Agonist, in Individuals with Renal Impairment: A Single-Dose, Phase I, Bridging Study.
저자
by
Klein, Gernot
;
Petrone, Marcella
;
Yang, Ye
;
Hoang, Thuong
;
Hazlett, Sheila
, et al.
소스
Clinical Pharmacokinetics
. Jun2023, Vol. 62 Issue 6, p881-890. 10p.
Web of Science
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7 . Academic Journal
Efficacy and safety of cotadutide, a dual glucagon‐like peptide‐1 and glucagon receptor agonist, in a randomized phase 2a study of patients with type 2 diabetes and chronic kidney disease.
저자
by
Parker, Victoria E. R.
;
Hoang, Thuong
;
Schlichthaar, Heike
;
Gibb, Fraser W.
;
Wenzel, Barbara
, et al.
소스
Diabetes, Obesity & Metabolism
. Jul2022, Vol. 24 Issue 7, p1360-1369. 10p.
Full Text (Wiley)
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7 . Academic Journal
A novel integrated QSP model of in vivo human glucose regulation to support the development of a glucagon/GLP‐1 dual agonist.
저자
by
Bosch, Rolien
;
Petrone, Marcella
;
Arends, Rosalin
;
Vicini, Paolo
;
Sijbrands, Eric J. G.
, et al.
소스
CPT: Pharmacometrics & Systems Pharmacology
. Mar2022, Vol. 11 Issue 3, p302-317. 16p.
Open Access (Wiley)
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7 . Academic Journal
Pharmacokinetics, safety, tolerability and efficacy of cotadutide, a glucagon‐like peptide‐1 and glucagon receptor dual agonist, in phase 1 and 2 trials in overweight or obese participants of Asian descent with or without type 2 diabetes.
저자
by
Asano, Michiko
;
Sekikawa, Akiko
;
Kim, Hyosung
;
Gasser, Robert A.
;
Robertson, Darren
, et al.
소스
Diabetes, Obesity & Metabolism
. Aug2021, Vol. 23 Issue 8, p1859-1867. 9p.
Full Text (Wiley)
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7 . Academic Journal
New fused benzazepine as selective D 3 receptor antagonists. Synthesis and biological evaluation. Part 2: [ g]-Fused and hetero-fused systems
저자
by
Micheli, Fabrizio
;
Bonanomi, Giorgio
;
Braggio, Simone
;
Capelli, Anna Maria
;
Damiani, Federica
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2008 18(3):908-912
Full Text (ScienceDirect)
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7 . Academic Journal
New fused benzazepine as selective D 3 receptor antagonists. Synthesis and biological evaluation. Part one: [h]-fused tricyclic systems
저자
by
Micheli, Fabrizio
;
Bonanomi, Giorgio
;
Braggio, Simone
;
Capelli, Anna Maria
;
Celestini, Paolo
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2008 18(3):901-907
Full Text (ScienceDirect)
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7 . Academic Journal
5-HT 2C antagonists based on fused heterotricyclic templates: Design, synthesis and biological evaluation
저자
by
Hamprecht, Dieter
;
Micheli, Fabrizio
;
Tedesco, Giovanna
;
Donati, Daniele
;
Petrone, Marcella
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2007 17(2):424-427
Full Text (ScienceDirect)
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7 . Academic Journal
Isoindolone derivatives, a new class of 5-HT 2C antagonists: Synthesis and biological evaluation
저자
by
Hamprecht, Dieter
;
Micheli, Fabrizio
;
Tedesco, Giovanna
;
Checchia, Anna
;
Donati, Daniele
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2007 17(2):428-433
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