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1 . Academic Journal
Design, synthesis, biological evaluation and crystal structure determination of dual modulators of carbonic anhydrases and estrogen receptors
저자
by
Tinivella, Annachiara
;
Nwachukwu, Jerome C.
;
Angeli, Andrea
;
Foschi, Francesca
;
Benatti, Anna Laura
, et al.
소스
In
European Journal of Medicinal Chemistry
15 January 2023 246
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7 . Academic Journal
Systems Structural Biology Analysis of Ligand Effects on ERα Predicts Cellular Response to Environmental Estrogens and Anti-hormone Therapies
저자
by
Nwachukwu, Jerome C.
;
Srinivasan, Sathish
;
Bruno, Nelson E.
;
Nowak, Jason
;
Wright, Nicholas J.
, et al.
소스
In
Cell Chemical Biology
19 January 2017 24(1):35-45
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7 . Academic Journal
The SARS-CoV-2 spike protein binds and modulates estrogen receptors.
저자
by
Solis, Oscar
;
Beccari, Andrea R.
;
Iaconis, Daniela
;
Talarico, Carmine
;
Ruiz-Bedoya, Camilo A.
, et al.
소스
Science Advances
. 12/2/2022, Vol. 8 Issue 48, p1-14. 14p.
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7 . Academic Journal
Unexpected equivalent potency of a constrained chromene enantiomeric pair rationalized by co-crystal structures in complex with estrogen receptor alpha
저자
by
Zhang, Birong
;
Kiefer, James R.
;
Blake, Robert A.
;
Chang, Jae H.
;
Hartman, Steven
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 April 2019 29(7):905-911
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7 . Academic Journal
Synthesis of novel steroidal agonists, partial agonists, and antagonists for the glucocorticoid receptor
저자
by
Jin, Zhuang
;
Lin, Hua
;
Srinivasan, Sathish
;
Nwachukwu, Jerome C.
;
Bruno, Nelson
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 January 2017 27(2):347-353
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7 . Periodical
Thiophene-Core Estrogen Receptor Ligands Having Superagonist Activity
저자
by
Min, Jian
;
Wang, Pengcheng
;
Srinivasan, Sathish
;
Nwachukwu, Jerome C.
;
Guo, Pu
, et al.
소스
Journal of Medicinal Chemistry; 20240101, Issue: Preprints
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7 . Periodical
Chemical systems biology reveals mechanisms of glucocorticoid receptor signaling
저자
by
Bruno, Nelson E.
;
Nwachukwu, Jerome C.
;
Srinivasan, Sathish
;
Nettles, Charles C.
;
Izard, Tina
, et al.
소스
Nature Chemical Biology; March 2021, Vol. 17 Issue: 3 p307-316, 10p
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7 . Academic Journal
Cryptic glucocorticoid receptor-binding sites pervade genomic NF-κB response elements.
저자
by
Hudson, William H.
;
de Vera, Ian Mitchelle S.
;
Nwachukwu, Jerome C.
;
Weikum, Emily R.
;
Herbst, Austin G.
, et al.
소스
Nature Communications; 4/6/2018, Vol. 9 Issue 1, p1-13, 13p, 4 Color Photographs, 1 Chart, 3 Graphs
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7 . Academic Journal
Tethering not required: the glucocorticoid receptor binds directly to activator protein-1 recognition motifs to repress inflammatory genes.
저자
by
Weikum, Emily R.
;
de Vera, Ian Mitchelle S.
;
Nwachukwu, Jerome C.
;
Hudson, William H.
;
Nettles, Kendall W.
, et al.
소스
Nucleic Acids Research; 8/21/2017, Vol. 45 Issue 14, p8596-8608, 13p
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7 . Periodical
Exploring the Structural Compliancy versus Specificity of the Estrogen Receptor Using Isomeric Three-Dimensional Ligands
저자
by
Sharma, Naina
;
Carlson, Kathryn E.
;
Nwachukwu, Jerome C.
;
Srinivasan, Sathish
;
Sharma, Abhishek
, et al.
소스
ACS Chemical Biology; February 2017, Vol. 12 Issue: 2 p494-503, 10p
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