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1 . Academic Journal
Lerisetron Analogues with Antimalarial Properties: Synthesis, Structure–Activity Relationship Studies, and Biological Assessment
저자
by
Rudolf Mueller
;
Virsinha Reddy
;
Aloysius T. Nchinda
;
Fanuel Mebrahtu
;
Dale Taylor
, et al.
소스
ACS Omega, Vol 5, Iss 12, Pp 6967-6982 (2020)
Open Access (DOAJ)
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7 . Academic Journal
Intestinal Transport Characteristics and Metabolism of C-Glucosyl Dihydrochalcone, Aspalathin
저자
by
Sandra Bowles
;
Elizabeth Joubert
;
Dalene de Beer
;
Johan Louw
;
Christel Brunschwig
, et al.
소스
Molecules, Vol 22, Iss 4, p 554 (2017)
Open Access (DOAJ)
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7 .
Novel 3-Trifluoromethyl-1,2,4-oxadiazole Analogues of Astemizole with Multi-stage Antiplasmodium Activity and In Vivo Efficacy in a Plasmodium berghei Mouse Malaria Infection Model
저자
by
Dickson Mambwe
;
Constance M. Korkor
;
Amanda Mabhula
;
Zama Ngqumba
;
Cleavon Cloete
, et al.
소스
Journal of Medicinal Chemistry
. 65:16695-16715
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7 .
1,3-Diarylpyrazolyl-acylsulfonamides as Potent Anti-tuberculosis Agents Targeting Cell Wall Biosynthesis in Mycobacterium tuberculosis
저자
by
Stephen Fienberg
;
Gregory S. Basarab
;
Anne J. Lenaerts
;
Virsinha Reddy
;
Sandeep R. Ghorpade
, et al.
소스
Journal of Medicinal Chemistry
. 64:12790-12807
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7 .
Benzoheterocyclic Oxime Carbamates Active against Mycobacterium tuberculosis: Synthesis, Structure–Activity Relationship, Metabolism, and Biology Triaging
저자
by
Ujjini H. Manjunatha
;
Christel Brunschwig
;
Mathew Njoroge
;
Srinivasa P. S. Rao
;
Nina Lawrence
, et al.
소스
Journal of Medicinal Chemistry
. 64:9444-9457
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7 .
Antimalarial Benzimidazole Derivatives Incorporating Phenolic Mannich Base Side Chains Inhibit Microtubule and Hemozoin Formation: Structure–Activity Relationship and In Vivo Oral Efficacy Studies
저자
by
Constance M. Korkor
;
Kelly Chibale
;
Godwin Akpeko Dziwornu
;
Sergio Wittlin
;
Dina Coertzen
, et al.
소스
Journal of Medicinal Chemistry
. 64:5198-5215
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7 .
Identification and Profiling of a Novel Diazaspiro[3.4]octane Chemical Series Active against Multiple Stages of the Human Malaria Parasite Plasmodium falciparum and Optimization Efforts
저자
by
Theresa L. Coetzer
;
Lizette L. Koekemoer
;
Elizabeth A. Winzeler
;
Gregory S. Basarab
;
Richard T. Eastman
, et al.
소스
Journal of Medicinal Chemistry
. 64:2291-2309
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7 .
New Amidated 3,6-Diphenylated Imidazopyridazines with Potent Antiplasmodium Activity Are Dual Inhibitors of Plasmodium Phosphatidylinositol-4-kinase and cGMP-Dependent Protein Kinase
저자
by
Sergio Wittlin
;
Lynn Wambua
;
Luyanda Centani
;
Lauren B. Arendse
;
Lyn-Marie Birkholtz
, et al.
소스
ACS Infectious Diseases
. 7:34-46
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7 .
Synthesis, Structure–Activity Relationship, and Mechanistic Studies of Aminoquinazolinones Displaying Antimycobacterial Activity
저자
by
Anthony J. Smith
;
Dale Taylor
;
Anne J. Lenaerts
;
Thomas R. Ioerger
;
Nina Lawrence
, et al.
소스
ACS Infectious Diseases
Open Access (OpenAIRE)
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7 .
Antitubercular 2-Pyrazolylpyrimidinones: Structure-Activity Relationship and Mode-of-Action Studies
저자
by
Kirsteen I. Buchanan
;
Clifton E. Barry
;
Simon Green
;
Gregory S. Basarab
;
Qin Su
, et al.
소스
Journal of Medicinal Chemistry
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