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1 . Academic Journal
Application of Imaging Mass Spectrometry to Assess Ocular Drug Transit
저자
by
Grove, Kerri J.
;
Kansara, Viral
;
Prentiss, Melissa
;
Long, Debby
;
Mogi, Muneto
, et al.
소스
In
SLAS Discovery
December 2017 22(10):1239-1245
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7 . Periodical
The Discovery of N-(1-Methyl-5-(trifluoromethyl)-1H-pyrazol-3-yl)-5-((6- ((methylamino)methyl)pyrimidin-4-yl)oxy)-1H-indole-1-carboxamide (Acrizanib), a VEGFR-2 Inhibitor Specifically Designed for Topical Ocular Delivery, as a Therapy for Neovascular Age-Related Macular Degeneration
저자
by
Adams, Christopher M.
;
Anderson, Karen
;
Artman, Gerald
;
Bizec, Jean-Claude
;
Cepeda, Rosemarie
, et al.
소스
Journal of Medicinal Chemistry; 20240101, Issue: Preprints
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7 . Academic Journal
The Discovery of N-(1-Methyl-5-(trifluoromethyl)-1H-pyrazol-3-yl)-5-((6- ((methylamino)methyl)pyrimidin-4-yl)oxy)-1H-indole-1-carboxamide (Acrizanib), a VEGFR-2 Inhibitor Specifically Designed for Topical Ocular Delivery, as a Therapy for Neovascular Age-Related Macular Degeneration.
저자
by
Adams, Christopher M.
;
Anderson, Karen
;
Artman Iii, Gerald
;
Bizec, Jean-Claude
;
Cepeda, Rosemarie
, et al.
소스
Journal of Medicinal Chemistry
. 2/22/2018, Vol. 61 Issue 4, p1622-1635. 14p.
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7 . Periodical
Discovery of 4-((2S,4S)-4-Ethoxy-1-((5-methoxy-7-methyl-1H-indol-4-yl)methyl)piperidin-2-yl)benzoic Acid (LNP023), a Factor B Inhibitor Specifically Designed To Be Applicable to Treating a Diverse Array of Complement Mediated Diseases
저자
by
Mainolfi, Nello
;
Ehara, Takeru
;
Karki, Rajeshri G.
;
Anderson, Karen
;
Mac Sweeney, Aengus
, et al.
소스
Journal of Medicinal Chemistry; June 2020, Vol. 63 Issue: 11 p5697-5722, 26p
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7 .
Phase I study of single agent NIZ985, a recombinant heterodimeric IL-15 agonist, in adult patients with metastatic or unresectable solid tumors
저자
by
Conlon, Kevin
;
Watson, Dionysios C
;
Waldmann, Thomas A
;
Valentin, Antonio
;
Bergamaschi, Cristina
, et al.
소스
Journal for Immunotherapy of Cancer
Journal for ImmunoTherapy of Cancer, Vol 9, Iss 11 (2021)
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7 . Periodical
Design, Synthesis, and Preclinical Characterization of Selective Factor D Inhibitors Targeting the Alternative Complement Pathway
저자
by
Karki, Rajeshri G.
;
Powers, James
;
Mainolfi, Nello
;
Anderson, Karen
;
Belanger, David B.
, et al.
소스
Journal of Medicinal Chemistry; April 2019, Vol. 62 Issue: 9 p4656-4668, 13p
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7 . Academic Journal
An EffectiveProdrug Strategy to Selectively EnhanceOcular Exposure of a Cannabinoid Receptor (CB1/2) Agonist.
저자
by
Mainolfi, Nello
;
Powers, James
;
Amin, Jakal
;
Long, Debby
;
Lee, Wendy
, et al.
소스
Journal of Medicinal Chemistry
. Vol. 56 Issue 13, p5464-5472. 9p.
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7 . Academic Journal
A topical VEGF inhibitor optimized for ocular indications
저자
by
Poor, Stephen H.
;
Adams, Christopher
;
Bigelow, Chad E.
;
Long, Debby
;
Yao, Penny
, et al.
소스
INVESTIGATIVE OPHTHALMOLOGY & VISUAL SCIENCE
; JUN 2017, 58 8, 4p.
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7 . Academic Journal
Pharmacologic Uncoupling of Angiogenesis and Inflammation during Initiation of Pathological Corneal Neovascularization.
저자
by
Sivak, Jeremy M.
;
Ostriker, Allison C.
;
Woolfenden, Amber
;
Demirs, John
;
Cepeda, Rosemarie
, et al.
소스
Journal of Biological Chemistry
. 12/30/2011, Vol. 286 Issue 52, p44965-44975. 11p.
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7 . Academic Journal
Long-acting protein drugs for the treatment of ocular diseases
저자
by
Ghosh, Joy G.
;
Nguyen, Andrew A.
;
Bigelow, Chad E.
;
Poor, Stephen
;
Qiu, Yubin
, et al.
소스
NATURE COMMUNICATIONS
; MAR 23 2017, 8 p14837 10p.
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