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1 . Academic Journal
Structural attributes influencing unbound tissue distribution
저자
by
Orozco, Christine C.
;
Atkinson, Karen
;
Ryu, Sangwoo
;
Chang, George
;
Keefer, Christopher
, et al.
소스
In
European Journal of Medicinal Chemistry
1 January 2020 185
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7 . Academic Journal
Modeling Exposure to Understand and Predict Kidney Injury
저자
by
Li, Zhenhong
;
Fisher, Ciaran
;
Gardner, Iain
;
Ghosh, Avijit
;
Litchfield, John
, et al.
소스
In
Seminars in Nephrology
March 2019 39(2):176-189
Full Text (ScienceDirect)
Full Text (Clinical Key)
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7 . Academic Journal
Development and evaluation of novel solid nanodispersion system for oral delivery of poorly water-soluble drugs
저자
by
Nkansah, Paul
;
Antipas, Amy
;
Lu, Ying
;
Varma, Manthena
;
Rotter, Charles
, et al.
소스
In
Journal of Controlled Release
10-28 July 2013 169(1-2):150-161
Full Text (ScienceDirect)
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7 . Academic Journal
Pharmacological inhibition of IRAK4 kinase activity does not prevent cachexia in mice with pancreatic cancer.
저자
by
Qiao, Shuxi
;
LaViolette, Brianna
;
Paulhus, Brianna LaCarubba
;
Li, Xiangping
;
Litchfield, John
, et al.
소스
JCSM Rapid Communications; Jul2023, Vol. 6 Issue 2, p122-133, 12p
Find it @ DONGA
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7 . Academic Journal
Target occupancy study and whole-body dosimetry with a MAGL PET ligand [
11
C]PF-06809247 in non-human primates.
저자
by
Arakawa, Ryosuke
;
Takano, Akihiro
;
Nag, Sangram
;
Jia, Zhisheng
;
Amini, Nahid
, et al.
소스
EJNMMI Research
. 3/4/2022, Vol. 12 Issue 1, p1-9. 9p.
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7 . Academic Journal
Identification of a novel conformationally constrained glucagon receptor antagonist
저자
by
Lee, Esther C.Y.
;
Tu, Meihua
;
Stevens, Benjamin D.
;
Bian, Jianwei
;
Aspnes, Gary
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 February 2014 24(3):839-844
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7 . Academic Journal
Metabolism of PF-04958242: Substrate concentration-dependent impact of cytochrome P4503A4 inhibitors as an explanation for a lack of clinical drug–drug interaction at very low substrate doses
저자
by
Obach, R. Scott
;
Doran, Angela C.
;
Shaffer, Christopher L.
;
Litchfield, John
.
소스
In
Drug Metabolism and Pharmacokinetics
January 2018 33(1) Supplement:S47-S47
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6 . Academic Journal
Effect of a Ketohexokinase Inhibitor (PF‐06835919) on In Vivo OATP1B Activity: Integrative Risk Assessment Using Endogenous Biomarker and a Probe Drug.
저자
by
Tess, David A.
;
Kimoto, Emi
;
King‐Ahmad, Amanda
;
Vourvahis, Manoli
;
Rodrigues, A. David
, et al.
소스
Clinical Pharmacology & Therapeutics; Sep2022, Vol. 112 Issue 3, p605-614, 10p
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7 . Academic Journal
Discovery of an intravenous hepatoselective glucokinase activator for the treatment of inpatient hyperglycemia
저자
by
Stevens, Benjamin D.
;
Litchfield, John
;
Pfefferkorn, Jeffrey A.
;
Atkinson, Karen
;
Perreault, Christian
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 December 2013 23(24):6588-6592
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7 . Academic Journal
Pyrimidone-based series of glucokinase activators with alternative donor–acceptor motif
저자
by
Filipski, Kevin J.
;
Guzman-Perez, Angel
;
Bian, Jianwei
;
Perreault, Christian
;
Aspnes, Gary E.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 August 2013 23(16):4571-4578
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