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1 . Academic Journal
Discovery, Optimization, and Biological Evaluation of Arylpyridones as Cbl‑b Inhibitors.
저자
by
Mfuh, Adelphe M.
;
Boerth, Jeffrey A.
;
Bommakanti, Gayathri
;
Chan, Christina
;
Chinn, Alex J.
, et al.
소스
Journal of Medicinal Chemistry; 1/25/2024, Vol. 67 Issue 2, p1500-1512, 13p
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7 . Academic Journal
Discovery of a Novel Benzodiazepine Series of Cbl‑b Inhibitors for the Enhancement of Antitumor Immunity.
저자
by
Boerth, Jeffrey A.
;
Chinn, Alex J.
;
Schimpl, Marianne
;
Bommakanti, Gayathri
;
Chan, Christina
, et al.
소스
ACS Medicinal Chemistry Letters; 12/14/2023, Vol. 14 Issue 12, p1848-1856, 9p
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7 . Academic Journal
AZD1208, a potent and selective pan-Pim kinase inhibitor, demonstrates efficacy in preclinical models of acute myeloid leukemia
저자
by
Keeton, Erika K.
;
McEachern, Kristen
;
Dillman, Keith S.
;
Palakurthi, Sangeetha
;
Cao, Yichen
, et al.
소스
In
Blood
6 February 2014 123(6):905-913
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7 . Academic Journal
Script-based automation of analytical instrument software tasks
저자
by
Tentarelli, Sharon
;
Romero, Rómulo
;
Lamb, Michelle L.
.
소스
In
SLAS Technology
June 2022 27(3):209-213
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5 . Academic Journal
Discovery and Optimization of the First ATP Competitive Type-III c‑MET Inhibitor.
저자
by
Michaelides, Iacovos N.
;
Collie, Gavin W.
;
Börjesson, Ulf
;
Vasalou, Christina
;
Alkhatib, Omar
, et al.
소스
Journal of Medicinal Chemistry; 7/13/2023, Vol. 66 Issue 13, p8782-8807, 26p
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7 . Academic Journal
Chapter 13 Targeting the Kinome with Computational Chemistry
저자
by
Lamb, Michelle L.
.
소스
In
Annual Reports in Computational Chemistry
2005 1:185-202
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3 . Academic Journal
Design of a gene family screening library targeting G-protein coupled receptors
저자
by
Lamb, Michelle L.
;
Bradley, Erin K.
;
Beaton, Graham
;
Bondy, Steven S.
;
Castellino, Angelo J.
, et al.
소스
In
Journal of Molecular Graphics and Modelling
2004 23(1):15-21
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7 . Academic Journal
Discovery of 2,6-disubstituted pyrazine derivatives as inhibitors of CK2 and PIM kinases
저자
by
Gingipalli, Lakshmaiah
;
Block, Michael H.
;
Bao, Larry
;
Cooke, Emma
;
Dakin, Les A.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 May 2018 28(8):1336-1341
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7 . Academic Journal
Mechanistic Insights into a CDK9 Inhibitor Via Orthogonal Proteomics Methods.
저자
by
Hendricks, J. Adam
;
Beaton, Nigel
;
Chernobrovkin, Alexey
;
Miele, Eric
;
Hamza, Ghaith M.
, et al.
소스
ACS Chemical Biology; 1/21/2022, Vol. 17 Issue 1, p54-67, 14p
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7 . Academic Journal
Modulating the strength of hydrogen bond acceptors to achieve low Caco2 efflux for oral bioavailability of PARP inhibitors blocking centrosome clustering
저자
by
Gu, Chungang
;
Lamb, Michelle L.
;
Johannes, Jeffrey W.
;
Sylvester, Mark A.
;
Eisman, Mark S.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 October 2016 26(19):4775-4780
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