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1 . Academic Journal
Phase I, Open-Label, Dose-Escalation Study of the Safety, Pharmacokinetics, Pharmacodynamics, and Efficacy of GSK2879552 in Relapsed/Refractory SCLC
저자
by
Bauer, Todd M.
;
Besse, Benjamin
;
Martinez-Marti, Alex
;
Trigo, Jose Manuel
;
Moreno, Victor
, et al.
소스
In
Journal of Thoracic Oncology
October 2019 14(10):1828-1838
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7 . Academic Journal
LSD1 inhibition exerts its antileukemic effect by recommissioning PU.1- and C/EBPα-dependent enhancers in AML
저자
by
Cusan, Monica
;
Cai, Sheng F.
;
Mohammad, Helai P.
;
Krivtsov, Andrei
;
Chramiec, Alan
, et al.
소스
In
Blood
12 April 2018 131(15):1730-1742
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7 . Academic Journal
EZH2 Is Required for Germinal Center Formation and Somatic EZH2 Mutations Promote Lymphoid Transformation
저자
by
Béguelin, Wendy
;
Popovic, Relja
;
Teater, Matt
;
Jiang, Yanwen
;
Bunting, Karen L.
, et al.
소스
In
Cancer Cell
13 May 2013 23(5):677-692
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7 . Academic Journal
Development and Validation of Reagents and Assays for EZH2 Peptide and Nucleosome High-Throughput Screens
저자
by
Diaz, Elsie
;
Machutta, Carl A.
;
Chen, Stephanie
;
Jiang, Yong
;
Nixon, Christopher
, et al.
소스
In
SLAS Discovery
December 2012 17(10):1279-1292
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7 . Academic Journal
Phase I trials of the lysine-specific demethylase 1 inhibitor, GSK2879552, as mono- and combination-therapy in relapsed/refractory acute myeloid leukemia or high-risk myelodysplastic syndromes.
저자
by
Roboz, Gail J.
;
Yee, Karen
;
Verma, Amit
;
Borthakur, Gautam
;
de la Fuente Burguera, Adolfo
, et al.
소스
Leukemia & Lymphoma
. Feb 2022, Vol. 63 Issue 2, p463-467. 5p.
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7 . Periodical
Fragment-based Scaffold Hopping: Identification of Potent, Selective, and Highly Soluble Bromo and Extra Terminal Domain (BET) Second Bromodomain (BD2) Inhibitors
저자
by
Seal, Jonathan T.
;
Atkinson, Stephen J.
;
Bamborough, Paul
;
Bassil, Anna
;
Chung, Chun-wa
, et al.
소스
Journal of Medicinal Chemistry; August 2021, Vol. 64 Issue: 15 p10772-10805, 34p
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7 . Academic Journal
LSD1 Inhibition Exerts Its Anti-Leukemic Effect By Recommissioning PU.1- and C/Ebpα-Dependent Enhancers in AML
저자
by
Cusan, Monica
;
Cai, Sheng
;
Mohammad, Helai P
;
Krivtsov, Andrei V.
;
Chramiec, Alan
, et al.
소스
In
Blood
8 December 2017 130 Supplement 1:242-242
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7 . Academic Journal
Discovery of a first-in-class reversible DNMT1-selective inhibitor with improved tolerability and efficacy in acute myeloid leukemia
저자
by
Pappalardi, Melissa B.
;
Keenan, Kathryn
;
Cockerill, Mark
;
Kellner, Wendy A.
;
Stowell, Alexandra
, et al.
소스
Nature Cancer
. 2(10):1002-1017
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7 . Academic Journal
Targeting Histone Methylation in Cancer
저자
by
McCabe, Michael T.
;
Mohammad, Helai P.
;
Barbash, Olena
;
Kruger, Ryan G.
.
소스
The Cancer Journal
. Sep 01, 2017 23(5):292-301
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6 .
In vitro and in vivo induction of fetal hemoglobin with a reversible and selective DNMT1 inhibitor
저자
by
Gilmartin, Aidan G.
;
Groy, Arthur
;
Gore, Elizabeth R.
;
Atkins, Charity
;
Long, Edward R.
, et al.
소스
Haematologica
Open Access (OpenAIRE)
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