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1 . Academic Journal
Natural product-inspired molecules for covalent inhibition of SHP2 tyrosine phosphatase
저자
by
Liang, Weida
;
Krabill, Aaron D.
;
Gallagher, Katelyn S.
;
Muli, Christine
;
Qu, Zihan
, et al.
소스
In
Tetrahedron
28 April 2024 156
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7 . Academic Journal
Altered Protein Dynamics and a More Reactive Catalytic Cysteine in a Neurodegeneration-associated UCHL1 Mutant
저자
by
Kenny, Sebastian
;
Lai, Chih-Hsuan
;
Chiang, Tsung-Sheng
;
Brown, Kwame
;
Hewitt, Chad S.
, et al.
소스
In
Journal of Molecular Biology
15 February 2024 436(4)
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7 . Academic Journal
Covalent Fragment Screening and Optimization Identifies the Chloroacetohydrazide Scaffold as Inhibitors for Ubiquitin C‑terminal Hydrolase L1.
저자
by
Imhoff, Ryan D.
;
Patel, Rishi
;
Safdar, Muhammad Hassan
;
Jones, Hannah B. L.
;
Pinto-Fernandez, Adan
, et al.
소스
Journal of Medicinal Chemistry; 3/28/2024, Vol. 67 Issue 6, p4496-4524, 29p
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7 . Academic Journal
Functional interrogation and therapeutic targeting of protein tyrosine phosphatases.
저자
by
Krabill, Aaron D.
;
Zhong-Yin Zhang
.
소스
Biochemical Society Transactions
. Aug2021, Vol. 49 Issue 4, p1723-1734. 12p.
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4 . Academic Journal
Development of Ubiquitin Variants with Selectivity for Ubiquitin C‑Terminal Hydrolase Deubiquitinases.
저자
by
Hewitt, Chad S.
;
Krabill, Aaron D.
;
Das, Chittaranjan
;
Flaherty, Daniel P.
.
소스
Biochemistry; 9/22/2020, Vol. 59 Issue 37, p3447-3462, 16p
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6 . Academic Journal
Optimization of Acetazolamide-Based Scaffold as Potent Inhibitors of Vancomycin-Resistant Enterococcus.
저자
by
Kaur, Jatinder
;
Cao, Xufeng
;
Abutaleb, Nader S.
;
Elkashif, Ahmed
;
Graboski, Amanda L.
, et al.
소스
Journal of Medicinal Chemistry; 9/10/2020, Vol. 63 Issue 17, p9540-9562, 23p
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7 . Academic Journal
Ubiquitin C‐Terminal Hydrolase L1: Biochemical and Cellular Characterization of a Covalent Cyanopyrrolidine‐Based Inhibitor.
저자
by
Krabill, Aaron D.
;
Chen, Hao
;
Hussain, Sajjad
;
Feng, Chao
;
Abdullah, Ammara
, et al.
소스
ChemBioChem; 3/2/2020, Vol. 21 Issue 5, p712-722, 11p
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7 . Academic Journal
Optimization and Anti-Cancer Properties of Fluoromethylketones as Covalent Inhibitors for Ubiquitin C-Terminal Hydrolase L1.
저자
by
Krabill, Aaron D.
;
Chen, Hao
;
Hussain, Sajjad
;
Hewitt, Chad S.
;
Imhoff, Ryan D.
, et al.
소스
Molecules
. Mar2021, Vol. 26 Issue 5, p1227-1227. 1p.
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7 . Academic Journal
Corrigendum: Ubiquitin C‐Terminal Hydrolase L1: Biochemical and Cellular Characterization of a Covalent Cyanopyrrolidine‐Based Inhibitor.
저자
by
Krabill, Aaron D.
;
Chen, Hao
;
Hussain, Sajjad
;
Feng, Chao
;
Abdullah, Ammara
, et al.
소스
ChemBioChem; 9/14/2020, Vol. 21 Issue 18, p2701-2701, 1p
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