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1 . Academic Journal
High throughput screening for compounds to the orphan nuclear receptor NR2F6
저자
by
Smith, Emery
;
Campbell, Sean
;
Wilson, Adrianna N.
;
Shumate, Justin
;
Baillargeon, Pierre
, et al.
소스
In
SLAS Discovery
June 2022 27(4):242-248
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7 . Academic Journal
Synthesis and structure activity relationship of the first class of LXR inverse agonists
저자
by
Elgendy, Bahaa
;
Griffett, Kristine
;
Hegazy, Lamees
;
Di Fruscia, Paolo
;
Sample, Kirby
, et al.
소스
In
Bioorganic Chemistry
February 2022 119
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7 . Academic Journal
PPARγ in Complex with an Antagonist and Inverse Agonist: a Tumble and Trap Mechanism of the Activation Helix
저자
by
Frkic, Rebecca L.
;
Marshall, Andrew C.
;
Blayo, Anne-Laure
;
Pukala, Tara L.
;
Kamenecka, Theodore M.
, et al.
소스
In
iScience
27 July 2018 5:69-79
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7 . Academic Journal
TNP [N2-(m-Trifluorobenzyl), N6-(p-nitrobenzyl)purine] ameliorates diet induced obesity and insulin resistance via inhibition of the IP6K1 pathway
저자
by
Ghoshal, Sarbani
;
Zhu, Qingzhang
;
Asteian, Alice
;
Lin, Hua
;
Xu, Haifei
, et al.
소스
In
Molecular Metabolism
October 2016 5(10):903-917
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7 . Academic Journal
Structure–Activity Relationship and Biological Investigation of a REV-ERBα-Selective Agonist SR-29065 (34) for Autoimmune Disorders.
저자
by
He, Yuanjun
;
Zhu, Di
;
Greenman, Kevin
;
Ruiz, Claudia
;
Shang, Jinsai
, et al.
소스
Journal of Medicinal Chemistry; 11/9/2023, Vol. 66 Issue 21, p14815-14823, 9p
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7 . Academic Journal
PPARγ Corepression Involves Alternate Ligand Conformation and Inflation of H12 Ensembles.
저자
by
Frkic, Rebecca L.
;
Pederick, Jordan L.
;
Horsfall, Aimee J.
;
Jovcevski, Blagojce
;
Crame, Elise E.
, et al.
소스
ACS Chemical Biology; 5/19/2023, Vol. 18 Issue 5, p1115-1123, 9p
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7 . Academic Journal
Identification of potent RORβ modulators: Scaffold variation
저자
by
Doebelin, Christelle
;
Patouret, Rémi
;
Garcia-Ordonez, Ruben D.
;
Chang, Mi Ra
;
Dharmarajan, Venkatasubramanian
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 October 2018 28(19):3210-3215
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7 . Academic Journal
Design, synthesis, and evaluation of simple phenol amides as ERRγ agonists
저자
by
Lin, Hua
;
Doebelin, Christelle
;
Patouret, Rémi
;
Garcia-Ordonez, Ruben D.
;
Chang, M.R.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 May 2018 28(8):1313-1319
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7 . Academic Journal
Identification of an aminothiazole series of RORβ modulators
저자
by
Patouret, Rémi
;
Doebelin, Christelle
;
Garcia-Ordonez, Ruben D.
;
Chang, Mi Ra
;
Ruiz, Claudia
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 April 2018 28(7):1178-1181
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7 . Academic Journal
Synthesis of novel steroidal agonists, partial agonists, and antagonists for the glucocorticoid receptor
저자
by
Jin, Zhuang
;
Lin, Hua
;
Srinivasan, Sathish
;
Nwachukwu, Jerome C.
;
Bruno, Nelson
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 January 2017 27(2):347-353
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