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1 . Academic Journal
A fluorescent splice-switching mouse model enables high-throughput, sensitive quantification of antisense oligonucleotide delivery and activity
저자
by
Byrnes, Amy E.
;
Roudnicky, Filip
;
Gogineni, Alvin
;
Soung, Allison L.
;
Xiong, Monica
, et al.
소스
In
Cell Reports Methods
22 January 2024 4(1)
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7 . Academic Journal
TMEM106B reduction does not rescue GRN deficiency in iPSC-derived human microglia and mouse models
저자
by
Dominguez, Sara L.
;
Laufer, Benjamin I.
;
Ghosh, Arundhati Sengupta
;
Li, Qingling
;
Ruggeri, Gaia
, et al.
소스
In
iScience
17 November 2023 26(11)
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7 . Academic Journal
Lipid nanoparticle delivery limits antisense oligonucleotide activity and cellular distribution in the brain after intracerebroventricular injection
저자
by
Byrnes, Amy E.
;
Dominguez, Sara L.
;
Yen, Chun-Wan
;
Laufer, Benjamin I.
;
Foreman, Oded
, et al.
소스
In
Molecular Therapy - Nucleic Acids
13 June 2023 32:773-793
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7 . Academic Journal
Anti-α-synuclein c-terminal antibodies block PFF uptake and accumulation of phospho-synuclein in preclinical models of Parkinson's disease
저자
by
Brendza, Robert
;
Gao, Xiaoying
;
Stark, Kimberly L.
;
Lin, Han
;
Lee, Seung-Hye
, et al.
소스
In
Neurobiology of Disease
February 2023 177
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7 . Academic Journal
Discovery of non-zwitterionic aryl sulfonamides as Nav1.7 inhibitors with efficacy in preclinical behavioral models and translational measures of nociceptive neuron activation
저자
by
Wu, Yong-Jin
;
Guernon, Jason
;
McClure, Andrea
;
Luo, Guanglin
;
Rajamani, Ramkumar
, et al.
소스
In
Bioorganic & Medicinal Chemistry
15 October 2017 25(20):5490-5505
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7 . Academic Journal
Triazolopyridine ethers as potent, orally active mGlu2 positive allosteric modulators for treating schizophrenia
저자
by
Higgins, Mendi A.
;
Marcin, Lawrence R.
;
Christopher Zusi, F.
;
Gentles, Robert
;
Ding, Min
, et al.
소스
In
Bioorganic & Medicinal Chemistry
15 January 2017 25(2):496-513
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7 . Academic Journal
Discovery of pyrrolo[2,1-f][1,2,4]triazine-based inhibitors of adaptor protein 2-associated kinase 1 for the treatment of pain.
저자
by
Dzierba, Carolyn D.
;
Dasgupta, Bireshwar
;
Karageorge, George
;
Kostich, Walter
;
Hamman, Brian
, et al.
소스
Medicinal Chemistry Research; Jul2023, Vol. 32 Issue 7, p1369-1375, 7p
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7 . Academic Journal
Difluorocyclobutylacetylenes as positive allosteric modulators of mGluR5 with reduced bioactivation potential
저자
by
Degnan, Andrew P.
;
Maxwell, Darrell
;
Balakrishnan, Anand
;
Brown, Jeffrey M.
;
Easton, Amy
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 December 2016 26(24):5871-5876
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7 . Academic Journal
Oxazolidinone-based allosteric modulators of mGluR5: Defining molecular switches to create a pharmacological tool box
저자
by
Huang, Hong
;
Degnan, Andrew P.
;
Balakrishnan, Anand
;
Easton, Amy
;
Gulianello, Michael
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 September 2016 26(17):4165-4169
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7 . Academic Journal
Acute Neurotoxicity of Antisense Oligonucleotides After Intracerebroventricular Injection Into Mouse Brain Can Be Predicted from Sequence Features.
저자
by
Hagedorn, Peter H.
;
Brown, Jeffrey M.
;
Easton, Amy
;
Pierdomenico, Maria
;
Jones, Kelli
, et al.
소스
Nucleic Acid Therapeutics
. Jun2022, Vol. 32 Issue 3, p151-162. 12p.
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