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1 . Academic Journal
Domain-selective targeting of BET proteins in cancer and immunological diseases
저자
by
Petretich, Massimo
;
Demont, Emmanuel H.
;
Grandi, Paola
.
소스
In
Current Opinion in Chemical Biology
August 2020 57:184-193
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5 . Academic Journal
Structure-Guided Design of a Domain-Selective Bromodomain and Extra Terminal N‑Terminal Bromodomain Chemical Probe.
저자
by
Bradley, Erin
;
Fusani, Lucia
;
Chung, Chun-wa
;
Craggs, Peter D.
;
Demont, Emmanuel H.
, et al.
소스
Journal of Medicinal Chemistry; 12/14/2023, Vol. 66 Issue 23, p15728-15749, 22p
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7 . Academic Journal
Design and Characterization of 1,3-Dihydro‑2H‑benzo[d]azepin-2-ones as Rule-of‑5 Compliant Bivalent BET Inhibitors.
저자
by
Bamborough, Paul
;
Chung, Chun-wa
;
Goodwin, Nicole C.
;
Mitchell, Darren J.
;
Neipp, Christopher E.
, et al.
소스
ACS Medicinal Chemistry Letters; 9/14/2023, Vol. 14 Issue 9, p1231-1236, 6p
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7 . Academic Journal
Multigram Synthesis of Tetrasubstituted Dihydrobenzofuran GSK973 Enabled by High-Throughput Experimentation and a Claisen Rearrangement in Flow.
저자
by
Alder, Catherine M.
;
Gray, Matthew
;
Huff, Chelsea A.
;
Manning, Calvin O.
;
Preston, Alex
, et al.
소스
Organic Process Research & Development; 2/18/2022, Vol. 26 Issue 2, p365-379, 15p
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7 . Academic Journal
Synthesis and structure–activity relationships of a series of (1 H-pyrazol-4-yl)acetamide antagonists of the P2X 7 receptor
저자
by
Chambers, Laura J.
;
Stevens, Alexander J.
;
Moses, Andrew P.
;
Michel, Anton D.
;
Walter, Daryl S.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2010 20(10):3161-3164
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7 . Periodical
Discovery of a Highly Selective BET BD2 Inhibitor from a DNA-Encoded Library Technology Screening Hit
저자
by
Rianjongdee, Francesco
;
Atkinson, Stephen J.
;
Chung, Chun-wa
;
Grandi, Paola
;
Gray, James R. J.
, et al.
소스
Journal of Medicinal Chemistry; August 2021, Vol. 64 Issue: 15 p10806-10833, 28p
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7 . Periodical
Fragment-based Scaffold Hopping: Identification of Potent, Selective, and Highly Soluble Bromo and Extra Terminal Domain (BET) Second Bromodomain (BD2) Inhibitors
저자
by
Seal, Jonathan T.
;
Atkinson, Stephen J.
;
Bamborough, Paul
;
Bassil, Anna
;
Chung, Chun-wa
, et al.
소스
Journal of Medicinal Chemistry; August 2021, Vol. 64 Issue: 15 p10772-10805, 34p
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7 . Periodical
Optimization of a Series of 2,3-Dihydrobenzofurans as Highly Potent, Second Bromodomain (BD2)-Selective, Bromo and Extra-Terminal Domain (BET) Inhibitors
저자
by
Lucas, Simon C. C.
;
Atkinson, Stephen J.
;
Chung, Chun-wa
;
Davis, Rob
;
Gordon, Laurie
, et al.
소스
Journal of Medicinal Chemistry; August 2021, Vol. 64 Issue: 15 p10711-10741, 31p
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7 . Academic Journal
Structure-Based Design of a Bromodomain and Extraterminal Domain (BET) Inhibitor Selective for the N‑Terminal Bromodomains That Retains an Anti-inflammatory and Antiproliferative Phenotype.
저자
by
Wellaway, Christopher R.
;
Bamborough, Paul
;
Bernard, Sharon G.
;
Chung, Chun-wa
;
Craggs, Peter D.
, et al.
소스
Journal of Medicinal Chemistry; 9/10/2020, Vol. 63 Issue 17, p9020-9044, 25p
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7 . Academic Journal
GSK789: A Selective Inhibitor of the First Bromodomains (BD1) of the Bromo and Extra Terminal Domain (BET) Proteins.
저자
by
Watson, Robert J.
;
Bamborough, Paul
;
Barnett, Heather
;
Chung, Chun-wa
;
Davis, Rob
, et al.
소스
Journal of Medicinal Chemistry; 9/10/2020, Vol. 63 Issue 17, p9045-9069, 25p
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