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1 . Academic Journal
Biomarker-driven strategy for MCL1 inhibition in T-cell lymphomas
저자
by
Koch, Raphael
;
Christie, Amanda L.
;
Crombie, Jennifer L.
;
Palmer, Adam C.
;
Plana, Deborah
, et al.
소스
In
Blood
7 February 2019 133(6):566-575
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7 . Academic Journal
A PKPD Case Study: Achieving Clinically Relevant Exposures of AZD5991 in Oncology Mouse Models.
저자
by
White, Michael J.
;
Cheatham, Letitia
;
Wen, Shenghua
;
Scarfe, Graeme
;
Cidado, Justin
, et al.
소스
AAPS Journal; Jul2023, Vol. 25 Issue 4, p1-8, 8p
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7 . Academic Journal
AZD4320 Is a Novel and Potent BCL-2/XL Dual Inhibitor in Targeting Aggressive Mantle Cell Lymphoma
저자
by
Li, Yijing
;
Liu, Yang
;
McIntosh, Joseph
;
Jordan, Alexa A
;
Leeming, Angela
, et al.
소스
In
Blood
5 November 2020 136 Supplement 1:44-44
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7 . Academic Journal
Sequential Inhibition of BCL-XL and MCL1 Elicits Massive Apoptosis in Anaplastic Thyroid Cancer Cells
저자
by
Shanja, Xhesika
;
Cidado, Justin
;
Di Cristofano, Antonio
.
소스
In
Journal of the American College of Surgeons
October 2020 231(4) Supplement 1:S80-S81
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5 . Academic Journal
Inhibition of Anti-Apoptotic Mcl-1 Exerts Anti-Leukemia Activity through Modulation of Leukemia-Stromal Interactions and Metabolic Functions in AML
저자
by
Carter, Bing Z
;
Mak, Po Yee
;
Warmoes, Marc
;
Tao, Wenjing
;
Lorenzi, Philip
, et al.
소스
In
Blood
13 November 2019 134 Supplement 1:3727-3727
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7 . Academic Journal
Combination of AZD4573, a Selective CDK9 Inhibitor, with Other Cell Death Inducing Agents Can Overcome De Novo Venetoclax Resistance in Preclinical Hematologic Tumor Models
저자
by
Cidado, Justin
;
Boiko, Scott
;
Proia, Theresa
;
Woods, Haley
;
Tavana, Omid
, et al.
소스
In
Blood
29 November 2018 132 Supplement 1:3946-3946
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7 . Academic Journal
Development and Use of Clinical Pharmacodynamic Assays to Demonstrate Target Engagement for AZD4573, a Selective and Potent CDK9 Inhibitor Currently in Phase I Clinical Trials
저자
by
Yeh, Tammie
;
O'Connor, Greg
;
Cidado, Justin
;
Barrett, J. Carl
.
소스
In
Blood
29 November 2018 132 Supplement 1:3505-3505
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6 .
Analysis of BRCA2 loss of heterozygosity in tumor tissue using droplet digital polymerase chain reaction
저자
by
Cochran, Rory L.
;
Cravero, Karen
;
Chu, David
;
Erlanger, Bracha
;
Toro, Patricia Valda
, et al.
소스
In
Human Pathology
July 2014 45(7):1546-1550
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7 . Academic Journal
Discovery of AZD4573, a Potent and Selective Inhibitor of CDK9 That Enables Short Duration of Target Engagement for the Treatment of Hematological Malignancies.
저자
by
Barlaam, Bernard
;
Casella, Robert
;
Cidado, Justin
;
Cook, Calum
;
De Savi, Chris
, et al.
소스
Journal of Medicinal Chemistry; 12/24/2020, Vol. 63 Issue 24, p15564-15590, 27p
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7 . Periodical
Targeting Bfl-1 via acute CDK9 inhibition overcomes intrinsic BH3-mimetic resistance in lymphomas
저자
by
Boiko, Scott
;
Proia, Theresa
;
San Martin, Maryann
;
Gregory, Gareth P.
;
Wu, Michelle Min
, et al.
소스
Blood; May 2021, Vol. 137 Issue: 21 p2947-2957, 11p
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