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1 . Academic Journal
Structure-guided optimization of 3-hydroxybenzoisoxazole derivatives as inhibitors of Aldo-keto reductase 1C3 (AKR1C3) to target prostate cancer
저자
by
Pippione, Agnese Chiara
;
Kovachka, Sandra
;
Vigato, Chiara
;
Bertarini, Laura
;
Mannella, Iole
, et al.
소스
In
European Journal of Medicinal Chemistry
15 March 2024 268
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7 . Academic Journal
Mechanisms of antiviral activity of the new hDHODH inhibitor MEDS433 against respiratory syncytial virus replication
저자
by
Luganini, Anna
;
Sibille, Giulia
;
Pavan, Marta
;
Mello Grand, Maurizia
;
Sainas, Stefano
, et al.
소스
In
Antiviral Research
November 2023 219
Full Text (ScienceDirect)
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7 . Academic Journal
Phenothiazines as anti-cancer agents: SAR overview and synthetic strategies
저자
by
Kumar, Arun
;
Vigato, Chiara
;
Boschi, Donatella
;
Lolli, Marco Lucio
;
Kumar, Deepak
.
소스
In
European Journal of Medicinal Chemistry
5 June 2023 254
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7 . Academic Journal
New aldo-keto reductase 1C3 (AKR1C3) inhibitors based on the hydroxytriazole scaffold
저자
by
Pippione, Agnese Chiara
;
Kilic-Kurt, Zühal
;
Kovachka, Sandra
;
Sainas, Stefano
;
Rolando, Barbara
, et al.
소스
In
European Journal of Medicinal Chemistry
5 July 2022 237
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7 . Academic Journal
Dihydroorotate dehydrogenase inhibitors in anti-infective drug research
저자
by
Boschi, Donatella
;
Pippione, Agnese Chiara
;
Sainas, Stefano
;
Lolli, Marco L.
.
소스
In
European Journal of Medicinal Chemistry
1 December 2019 183
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6 . Academic Journal
CML-164 Dihydroorotate Dehydrogenase Inhibition Reveals Metabolic Vulnerability in Chronic Myeloid Leukemia
저자
by
Houshmand, Mohammad
;
Vitale, Nicoletta
;
Orso, Francesca
;
Cignetti, Alessandro
;
Molineris, Ivan
, et al.
소스
In
Clinical Lymphoma, Myeloma and Leukemia
October 2022 22 Supplement 2:S288-S289
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7 . Academic Journal
Hydroxyazole scaffold-based Plasmodium falciparum dihydroorotate dehydrogenase inhibitors: Synthesis, biological evaluation and X-ray structural studies
저자
by
Pippione, Agnese C.
;
Sainas, Stefano
;
Goyal, Parveen
;
Fritzson, Ingela
;
Cassiano, Gustavo C.
, et al.
소스
In
European Journal of Medicinal Chemistry
1 February 2019 163:266-280
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7 . Academic Journal
4-Hydroxy-1,2,3-triazole moiety as bioisostere of the carboxylic acid function: a novel scaffold to probe the orthosteric γ-aminobutyric acid receptor binding site
저자
by
Giraudo, Alessandro
;
Krall, Jacob
;
Nielsen, Birgitte
;
Sørensen, Troels E.
;
Kongstad, Kenneth T.
, et al.
소스
In
European Journal of Medicinal Chemistry
5 October 2018 158:311-321
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7 . Academic Journal
Potent and selective aldo-keto reductase 1C3 (AKR1C3) inhibitors based on the benzoisoxazole moiety: application of a bioisosteric scaffold hopping approach to flufenamic acid
저자
by
Pippione, Agnese Chiara
;
Carnovale, Irene Maria
;
Bonanni, Davide
;
Sini, Marcella
;
Goyal, Parveen
, et al.
소스
In
European Journal of Medicinal Chemistry
25 April 2018 150:930-945
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7 . Academic Journal
Hydroxytriazole derivatives as potent and selective aldo-keto reductase 1C3 (AKR1C3) inhibitors discovered by bioisosteric scaffold hopping approach
저자
by
Pippione, Agnese C.
;
Giraudo, Alessandro
;
Bonanni, Davide
;
Carnovale, Irene M.
;
Marini, Elisabetta
, et al.
소스
In
European Journal of Medicinal Chemistry
20 October 2017 139:936-946
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