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1 . Academic Journal
Design, Synthesis, and Characterization of I-BET567, a Pan-Bromodomain and Extra Terminal (BET) Bromodomain Oral Candidate.
저자
by
Humphreys, Philip G.
;
Atkinson, Stephen J.
;
Bamborough, Paul
;
Bit, Rino A.
;
Chun-wa Chung
, et al.
소스
Journal of Medicinal Chemistry; 2/10/2022, Vol. 65 Issue 3, p2262-2287, 26p
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7 . Academic Journal
Pyrazolopyridazine alpha-2-delta-1 ligands for the treatment of neuropathic pain
저자
by
Myatt, James W.
;
Healy, Mark P.
;
Bravi, Gianpaolo S.
;
Billinton, Andrew
;
Johnson, Christopher N.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 August 2010 20(15):4683-4688
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7 . Academic Journal
Novel methylene-linked heterocyclic EP 1 receptor antagonists
저자
by
Hall, Adrian
;
Bit, Rino A.
;
Brown, Susan H.
;
Chowdhury, Anita
;
Giblin, Gerard M.P.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2008 18(5):1592-1597
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7 . Academic Journal
The discovery of 6-[2-(5-chloro-2-{[(2,4-difluorophenyl)methyl]oxy}phenyl)-1-cyclopenten-1-yl]-2-pyridinecarboxylic acid, GW848687X, a potent and selective prostaglandin EP 1 receptor antagonist for the treatment of inflammatory pain
저자
by
Giblin, Gerard M.P.
;
Bit, Rino A.
;
Brown, Susan H.
;
Chaignot, Hélène M.
;
Chowdhury, Anita
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2007 17(2):385-389
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7 . Academic Journal
Discovery of novel biaryl heterocyclic EP1 receptor antagonists
저자
by
Hall, Adrian
;
Bit, Rino A.
;
Brown, Susan H.
;
Chaignot, Helene M.
;
Chessell, Iain P.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 May 2006 16(10):2666-2671
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7 . Periodical
Discovery of a Bromodomain and Extraterminal Inhibitor with a Low Predicted Human Dose through Synergistic Use of Encoded Library Technology and Fragment Screening
저자
by
Wellaway, Christopher R.
;
Amans, Dominique
;
Bamborough, Paul
;
Barnett, Heather
;
Bit, Rino A.
, et al.
소스
Journal of Medicinal Chemistry; January 2020, Vol. 63 Issue: 2 p714-746, 33p
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7 . Academic Journal
Structure-based design of peptidomimetic antagonists of p56 lck SH2 Domain
저자
by
Hobbs, Christopher J.
;
Bit, Rino A.
;
Cansfield, Andrew D.
;
Harris, Bill
;
Hill, Christopher H.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2002 12(10):1365-1369
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7 . Academic Journal
Discovery of I-BRD9, a Selective Cell Active Chemical Probe for Bromodomain Containing Protein 9 Inhibition.
저자
by
Theodoulou, Natalie H.
;
Bamborough, Paul
;
Bannister, Andrew J.
;
Becher, Isabelle
;
Bit, Rino A.
, et al.
소스
Journal of Medicinal Chemistry
. Feb2016, Vol. 59 Issue 4, p1425-1439. 15p.
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7 . Academic Journal
Discovery of Tetrahydropyrazolopyridine as Sphingosine 1-Phosphate Receptor 3 (S1P
3
)-Sparing S1P
1
Agonists Active at Low Oral Doses.
저자
by
Demont, Emmanuel H.
;
Bailey, James M.
;
Bit, Rino A.
;
Brown, Jack A.
;
Campbell, Colin A.
, et al.
소스
Journal of Medicinal Chemistry
. Feb2016, Vol. 59 Issue 3, p1003-1020. 18p.
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7 . Academic Journal
Optimization of Sphingosine-1-phosphate-1ReceptorAgonists: Effects of Acidic, Basic, and Zwitterionic Chemotypes onPharmacokinetic and Pharmacodynamic Profiles.
저자
by
Skidmore, John
;
Heer, Jag
;
Johnson, Christopher N.
;
Norton, David
;
Redshaw, Sally
, et al.
소스
Journal of Medicinal Chemistry
. Dec2014, Vol. 57 Issue 24, p10424-10442. 19p.
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