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1 . Academic Journal
Novel Indane-Containing NBTIs with Potent Anti-Gram-Negative Activity and Minimal hERG Inhibition.
저자
by
Cumming, John G.
;
Kreis, Lukas
;
Kühne, Holger
;
Wermuth, Roger
;
Vercruysse, Maarten
, et al.
소스
ACS Medicinal Chemistry Letters; 12/14/2023, Vol. 14 Issue 12, p1791-1799, 9p
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7 . Academic Journal
Structure-guided design of antibacterials that allosterically inhibit DNA gyrase
저자
by
Thalji, Reema K.
;
Raha, Kaushik
;
Andreotti, Daniele
;
Checchia, Anna
;
Cui, Haifeng
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 June 2019 29(11):1407-1412
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7 . Academic Journal
Synthesis of new polysubstituted piperazines and dihydro-2 H-pyrazines by selective reduction of 2-oxo-piperazines
저자
by
Reginato, Gianna
;
Credico, Barbara Di
;
Andreotti, Daniele
;
Mingardi, Anna
;
Paio, Alfredo
, et al.
소스
In
Tetrahedron: Asymmetry
2010 21(2):191-194
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7 . Academic Journal
A new versatile and diastereoselective synthesis of polysubstituted 2-oxopiperazines from naturally occurring amino acids
저자
by
Reginato, Gianna
;
Di Credico, Barbara
;
Andreotti, Daniele
;
Mingardi, Anna
;
Paio, Alfredo
, et al.
소스
In
Tetrahedron: Asymmetry
2007 18(22):2680-2688
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7 . Academic Journal
Discovery of 5-substituent-N-arylbenzamide derivatives as potent, selective and orally bioavailable LRRK2 inhibitors
저자
by
Ding, Xiao
;
Dai, Xuedong
;
Long, Kai
;
Peng, Cheng
;
Andreotti, Daniele
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 September 2017 27(17):4034-4038
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7 . Academic Journal
GSK2578215A; A potent and highly selective 2-arylmethyloxy-5-substitutent-N-arylbenzamide LRRK2 kinase inhibitor
저자
by
Reith, Alastair D.
;
Bamborough, Paul
;
Jandu, Karamjit
;
Andreotti, Daniele
;
Mensah, Lucy
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 September 2012 22(17):5625-5629
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7 . Academic Journal
Mechanism insights into an unexpected isomerisation reaction observed during conversion of N-benzyl piperazinones to corresponding N-benzyl thio-piperazinones
저자
by
Miserazzi, Emanuele
;
Spotti, Mario Alessandro
;
Profeta, Roberto
;
Spada, Simone
;
Nalin, Arnaldo
, et al.
소스
In
Tetrahedron Letters
19 January 2011 52(3):448-452
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7 . Academic Journal
A specific and direct comparison of the trifluoromethyl and pentafluoro sulfanyl groups on the selective dopamine D3 antagonist 3-(3-{[4-methyl-5-(4-methyl-1,3-oxazol-5-yl)-4H-1,2,4-triazol-3-yl]thio}propyl)-1-phenyl-3-azabicyclo[3.1.0]hexane template
저자
by
Micheli, Fabrizio
;
Andreotti, Daniele
;
Braggio, Simone
;
Checchia, Anna
.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 August 2010 20(15):4566-4568
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6 . Periodical
Discovery of N-[(2S)-5-(6-Fluoro-3-pyridinyl)-2,3-dihydro-1H-inden-2-yl]-2-propanesulfonamide, a Novel Clinical AMPA Receptor Positive Modulator
저자
by
Ward, Simon E.
;
Harries, Mark
;
Aldegheri, Laura
;
Andreotti, Daniele
;
Ballantine, Stuart
, et al.
소스
Journal of Medicinal Chemistry; 20240101, Issue: Preprints
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7 . Academic Journal
Selective Inhibitors of G2019S-LRRK2 Kinase Activity.
저자
by
Garofalo, Albert W.
;
Bright, Jessica
;
De Lombaert, Stéphane
;
Toda, Alyssa M. A.
;
Zobel, Kerry
, et al.
소스
Journal of Medicinal Chemistry; 12/10/2020, Vol. 63 Issue 23, p14821-14839, 19p
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