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1 .
Scaffold morphing leading to evolution of 2,4-diaminoquinolines and aminopyrazolopyrimidines as inhibitors of the ATP synthesis pathway
저자
by
Manoranjan Panda
;
Anandkumar Raichurkar
;
Neela Dinesh
;
Vinayak Hosagrahara
;
Naveen Kumar
, et al.
소스
MedChemComm
. 7:1022-1032
Scopus
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7 .
Novel lead generation of an anti-tuberculosis agent active against non-replicating mycobacteria: exploring hybridization of pyrazinamide with multiple fragments
저자
by
Parvinder Kaur
;
Shankar D. Markad
;
B. K. Kishore Reddy
;
Manoranjan Panda
;
Murugan Chinnapattu
, et al.
소스
Medicinal Chemistry Research
. 24:2986-2992
Web of Science
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7 .
Structure Guided Lead Generation for M. tuberculosis Thymidylate Kinase (Mtb TMK): Discovery of 3-Cyanopyridone and 1,6-Naphthyridin-2-one as Potent Inhibitors
저자
by
Rajesh Kalkhambkar
;
Bheemarao G. Ugarkar
;
Jon Read
;
Martin Vogtherr
;
Beena Paul
, et al.
소스
Journal of Medicinal Chemistry
. 58:753-766
Web of Science
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7 .
Benzimidazoles: Novel Mycobacterial Gyrase Inhibitors from Scaffold Morphing
저자
by
Jitendar Reddy
;
Parvinder Kaur
;
Dharmarajan Sriram
;
Anandkumar Raichurkar
;
Sreevalli Sharma
, et al.
소스
ACS Medicinal Chemistry Letters
. 5:820-825
Open Access (OpenAIRE)
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7 .
Shared Consensus Machine Learning Models for Predicting Blood Stage Malaria Inhibition
저자
by
Thierry Kogej
;
Chris L. Waller
;
Darren V. S. Green
;
Anandkumar Raichurkar
;
George Papadatos
, et al.
소스
Journal of chemical information and modeling
. 57(3)
Scopus
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7 .
Novel N-Linked Aminopiperidine-Based Gyrase Inhibitors with Improved hERG and in Vivo Efficacy against Mycobacterium tuberculosis
저자
by
V. K. Ramya
;
Vijender Panduga
;
Gajanan Shanbhag
;
Michelle Coulson
;
Sowmya Bharath
, et al.
소스
Journal of Medicinal Chemistry
. 57:4889-4905
Web of Science
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7 .
Discovery of Pyrazolopyridones as a Novel Class of Noncovalent DprE1 Inhibitor with Potent Anti-Mycobacterial Activity
저자
by
Parvinder Kaur
;
Anisha Ambady
;
Sreevalli Sharma
;
Vinayak Hosagrahara
;
Ashwini Narayan
, et al.
소스
Journal of Medicinal Chemistry
. 57:4761-4771
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7 .
Thiazolopyridone ureas as DNA gyrase B inhibitors: Optimization of antitubercular activity and efficacy
저자
by
P. Ann Boriack-Sjodin
;
B. K. Kishore Reddy
;
Ramesh R. Kale
;
Vijaykamal Ahuja
;
Sunita M. de Sousa
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 24:870-879
Web of Science
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7 .
Left-Hand Side Exploration of Novel Bacterial Topoisomerase Inhibitors to Improve Selectivity against hERG Binding
저자
by
Suresh Rudrapatana
;
Anandkumar Raichurkar
;
Vasan K. Sambandamurthy
;
Vikas Shinde
;
Sreevalli Sharma
, et al.
소스
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7 .
Triaminopyrimidine is a fast-killing and long-acting antimalarial clinical candidate
저자
by
Shridhar Narayanan
;
Laura M. Sanz
;
Sreenivasaiah Menasinakai
;
Kevin Hickling
;
Abhishek Srivastava
, et al.
소스
Nature Communications
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