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41 .
A phase I dose escalation, safety and pharmacokinetic (PK) study of AZD5312 (IONIS-ARRx), a first-in-class Generation 2.5 antisense oligonucleotide targeting the androgen receptor (AR)
저자
by
H.-T. Arkenau
;
T. Coleman
;
M. Voskoboynik
;
J. R. Infante
;
H. Gardner
, et al.
소스
European Journal of Cancer
. 69:S145
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47 .
AZD1208, a potent and selective pan-Pim kinase inhibitor, demonstrates efficacy in preclinical models of acute myeloid leukemia
저자
by
Yichen Cao
;
Surinder Kaur
;
Paul Lyne
;
Dennis Huszar
;
Suping Wang
, et al.
소스
Blood
. 123(6)
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47 .
501 Immunological STAT3 knockdown associated with anti-tumor activity in pre-clinical models translates to clinical samples, suggesting immune modulation contributes to the clinical activity of AZD9150, a therapeutic STAT3 ASO
저자
by
David S. Hong
;
C.C. Lin
;
Corinne Reimer
;
Michael Collins
;
Y.K. Kang
, et al.
소스
European Journal of Cancer
. 50:163-164
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47 .
Discovery and optimization of a novel series of potent mutant B-Raf(V600E) selective kinase inhibitors
저자
by
Charles A. Omer
;
Donald N. Cook
;
Jeffrey W. Johannes
;
Lisa Drew
;
Timothy Pontz
, et al.
소스
Journal of medicinal chemistry
. 56(5)
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47 .
Abstract 4705: Therapeutic activity of bivalent BRD4 inhibitor AZD5153 in hematological cancers
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by
Huawei (Ray) Chen
;
Maureen Hattersley
;
Garrett Rhyasen
;
Austin Dulak
;
Wendy Wang
, et al.
소스
Cancer Research
. 76:4705-4705
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47 .
Abstract 1971: BRD4 amplification facilitates an oncogenic gene expression program in high-grade serous ovarian cancer
저자
by
Garrett W. Rhyasen
;
Stephen E. Fawell
;
Paul Lyne
;
Michael Zinda
;
Maureen Hattersley
, et al.
소스
Cancer Research
. 76:1971-1971
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47 .
Discovery of Disubstituted Imidazo[4,5-b]pyridines and Purines as Potent TrkA Inhibitors
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by
Hai-Jun Zhang
;
Paul Lyne
;
Ethan Hoffmann
;
Dingwei Yu
;
Michael Howard Block
, et al.
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47 .
Discovery of checkpoint kinase inhibitor (S)-5-(3-fluorophenyl)-N-(piperidin-3-yl)-3-ureidothiophene-2-carboxamide (AZD7762) by structure-based design and optimization of thiophenecarboxamide ureas
저자
by
Siân Rowsell
;
Shannon Ready
;
James W. Janetka
;
Dongfang Liu
;
Paul Lyne
, et al.
소스
Journal of medicinal chemistry
. 55(11)
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47 .
Discovery of novel benzylidene-1,3-thiazolidine-2,4-diones as potent and selective inhibitors of the PIM-1, PIM-2, and PIM-3 protein kinases
저자
by
James E. Dowling
;
Michelle Lamb
;
Erika Krasnickas Keeton
;
Alexander Hird
;
Erin Code
, et al.
소스
Bioorganicmedicinal chemistry letters
. 22(14)
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47 .
Abstract PR12: Discovery and preclinical evaluation of cEt-modified KRAS antisense oligonucleotide inhibitors
저자
by
Brett P. Monia
;
Sarah Ross
;
Mitchell Revill
;
Stephanie Klein
;
Alexey S. Revenko
, et al.
소스
Molecular Cancer Therapeutics
. 14:PR12-PR12
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