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21 . Academic Journal
Utility of Resazurin, Horseradish Peroxidase, and NMR Assays to Identify Redox-Related False-Positive Behavior in High-Throughput Screens.
저자
by
Tarnowski, Matthew
;
Barozet, Amélie
;
Johansson, Carina
;
Eriksson, Per-Olof
;
Engkvist, Ola
, et al.
소스
Assay & Drug Development Technologies; Apr2018, Vol. 16 Issue 3, p171-191, 15p
Web of Science
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27 . Periodical
Seven Year Itch: Pan-Assay Interference Compounds (PAINS) in 2017Utility and Limitations
저자
by
Baell, Jonathan B.
;
Nissink, J. Willem M.
.
소스
ACS Chemical Biology; December 2017, Vol. 13 Issue: 1 p36-44, 9p
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24 . Academic Journal
Potent and Selective Inhibitors of MTH1 Probe Its Role in Cancer Cell Survival.
저자
by
Kettle, Jason G.
;
Alwan, Husam
;
Bista, Michal
;
Breed, Jason
;
Davies, Nichola L.
, et al.
소스
Journal of Medicinal Chemistry
. Mar2016, Vol. 59 Issue 6, p2346-2361. 16p.
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27 . Academic Journal
MTH1 Substrate Recognition—An Example of Specific Promiscuity.
저자
by
Nissink, J. Willem M.
;
Bista, Michal
;
Breed, Jason
;
Carter, Nikki
;
Embrey, Kevin
, et al.
소스
PLoS ONE
. 3/21/2016, Vol. 11 Issue 3, p1-16. 16p.
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27 . Periodical
Discovery of a Potent and Orally Bioavailable Zwitterionic Series of Selective Estrogen Receptor Degrader-Antagonists
저자
by
Scott, James S.
;
Stead, Darren
;
Barlaam, Bernard
;
Breed, Jason
;
Carbajo, Rodrigo J.
, et al.
소스
Journal of Medicinal Chemistry; 20230101, Issue: Preprints
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27 . Academic Journal
PAINS in the Assay: Chemical Mechanisms of Assay Interference and Promiscuous Enzymatic Inhibition Observed during a Sulfhydryl-Scavenging HTS.
저자
by
Dahlin, Jayme L.
;
Nissink, J. Willem M.
;
Strasser, Jessica M.
;
Francis, Subhashree
;
Higgins, LeeAnn
, et al.
소스
Journal of Medicinal Chemistry
. Mar2015, Vol. 58 Issue 5, p2091-2113. 23p.
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27 . Academic Journal
Promiscuous 2-Aminothiazoles(PrATs): A FrequentHitting Scaffold.
저자
by
Devine, Shane M.
;
Mulcair, Mark D.
;
Debono, Cael O.
;
Leung, Eleanor W. W.
;
Nissink, J. Willem M.
, et al.
소스
Journal of Medicinal Chemistry
. Feb2015, Vol. 58 Issue 3, p1205-1214. 10p.
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27 . Academic Journal
Analyzing compound and project progress through multi-objective-based compound quality assessment.
저자
by
Nissink, J. Willem M.
;
Degorce, Sébastien
.
소스
Future Medicinal Chemistry; Jun2013, Vol. 5 Issue 7, p753-767, 15p
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24 . Academic Journal
Discovery of 4‑{4-[(3R)‑3-Methylmorpholin-4-yl]-6-[1-(methylsulfonyl)cyclopropyl]pyrimidin-2-yl}‑1H‑indole (AZ20): A Potent and Selective Inhibitor of ATR Protein Kinase with Monotherapy in Vivo Antitumor Activity.
저자
by
Foote, Kevin M.
;
Blades, Kevin
;
Cronin, Anna
;
Fillery, Shaun
;
Guichard, Sylvie S.
, et al.
소스
Journal of Medicinal Chemistry
. 3/14/2013, Vol. 56 Issue 5, p2125-2138. 14p.
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27 . Academic Journal
Structures of the Human Poly (ADP-Ribose) Glycohydrolase Catalytic Domain Confirm Catalytic Mechanism and Explain Inhibition by ADP-HPD Derivatives.
저자
by
Tucker, Julie A.
;
Bennett, Neil
;
Brassington, Claire
;
Durant, Stephen T.
;
Hassall, Giles
, et al.
소스
PLoS ONE
. Dec2012, Vol. 7 Issue 12, p1-19. 19p.
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