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21 .
Unravelling the Turn‐On Fluorescence Mechanism of a Fluorescein‐Based Probe in GABA A Receptors
저자
by
Pedro Alejandro Sánchez-Murcia
;
Margot Ernst
;
Leticia Gonzalez
;
Nadja Katharina Singer
.
소스
Angewandte Chemie
. 134
Full Text (Wiley)
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26 .
A de novo missense variant in GABRA4 alters receptor function in an epileptic and neurodevelopmental phenotype
저자
by
Florian D. Vogel
;
Martin Krenn
;
Dominik S. Westphal
;
Elisabeth Graf
;
Matias Wagner
, et al.
소스
Epilepsia 63, e35-e41 (2022)
Open Access (OpenAIRE)
Scopus
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27 .
A Benzodiazepine Ligand with Improved GABAA Receptor α5-Subunit Selectivity Driven by Interactions with Loop C
저자
by
Petra Scholze
;
Roshan Puthenkalam
;
Margot Ernst
;
Markus Müllegger
;
Xenia Simeone
, et al.
소스
Molecular Pharmacology
. 99:39-48
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27 .
GABA A Receptor Modulators
저자
by
Luca L Silva
;
Margot Ernst
;
Florian Vogel
.
소스
eLS
. :1-10
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25 .
Variations on a scaffold - Novel GABAA receptor modulators
저자
by
Berthold Stoeger
;
Margot Ernst
;
Maria Teresa Iorio
;
Michael Schnürch
;
Sabah Rehman
, et al.
소스
European Journal of Medicinal Chemistry
. 180:340-349
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27 .
Phenotypic variability of GABRA1 ‐related epilepsy in monozygotic twins
저자
by
Fritz Zimprich
;
Matias Wagner
;
Martin Krenn
;
Margot Ernst
;
Thomas Meitinger
, et al.
소스
Annals of Clinical and Translational Neurology
Ann. Clin. Transl. Neurol. 6, 2317-2322 (2019)
Annals of Clinical and Translational Neurology, Vol 6, Iss 11, Pp 2317-2322 (2019)
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27 .
Defined concatenated α6α1β3γ2 GABAA receptor constructs reveal dual action of pyrazoloquinolinone allosteric modulators
저자
by
Margot Ernst
;
Sabah Rehman
;
Marko D. Mihovilovic
;
Xenia Simeone
;
Michael Schnürch
, et al.
소스
Bioorganic & Medicinal Chemistry
. 27:3167-3178
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27 .
The α6 subunit-containing GABAA receptor: A novel drug target for inhibition of trigeminal activation
저자
by
Pi-Chuan Fan
;
Pokai Huang
;
Lih-Chu Chiou
;
Chia Chun Hor
;
Daniel E. Knutson
, et al.
소스
Neuropharmacology
. 140:1-13
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27 .
Attaining in vivo selectivity of positive modulation of α3βγ2 GABAA receptors in rats: A hard task!
저자
by
Margot Ernst
;
Veera Venkata Naga Phani Babu Tiruveedhula
;
Aleksandar Obradovic
;
Miroslav M. Savić
;
Tamara Stankovic
, et al.
소스
European Neuropsychopharmacology
. 28:903-914
Full Text (Clinical Key)
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27 .
SAR-Guided Scoring Function and Mutational Validation Reveal the Binding Mode of CGS-8216 at the α1+/γ2– Benzodiazepine Site
저자
by
Marcus Wieder
;
Gerhard F. Ecker
;
Margot Ernst
;
Marko D. Mihovilovic
;
Thierry Langer
, et al.
소스
Journal of Chemical Information and Modeling
. 58:1682-1696
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