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21 . Academic Journal
Structural and signaling mechanisms of TAAR1 enabled preferential agonist design
저자
by
Shang, Pan
;
Rong, Naikang
;
Jiang, Jing-Jing
;
Cheng, Jie
;
Zhang, Ming-Hui
, et al.
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Cell
22 November 2023 186(24):5347-5362
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27 . Academic Journal
5-Cyano substituted diarylpyridines as potent HIV-1 NNRTIs: Rational design, synthesis, and activity evaluation
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by
Song, Hao
;
Xia, Yu
;
Zhang, Tao
;
Dun, Caiyun
;
Meng, Bairu
, et al.
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European Journal of Medicinal Chemistry
5 November 2023 259
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27 . Academic Journal
Medicinal chemistry strategies in the discovery and optimization of HBV core protein allosteric modulators (2018–2022 update)
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by
Shao, Xiaoyu
;
Xu, Shujing
;
Wan, Xufeng
;
Zhou, Yang
;
Wang, Shuo
, et al.
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Chinese Chemical Letters
November 2023 34(11)
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27 . Academic Journal
Discovery of novel diarypyrimidine derivatives bearing six-membered non-aromatic heterocycles as potent HIV-1 NNRTIs with improved anti-resistance and drug-like profiles
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by
Jiang, Xiangyi
;
Huang, Boshi
;
Zalloum, Waleed A.
;
Chen, Chin-Ho
;
Ji, Xiangkai
, et al.
소스
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European Journal of Medicinal Chemistry
5 October 2023 258
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27 . Academic Journal
Targeting hepatitis B virus cccDNA levels: Recent progress in seeking small molecule drug candidates
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by
Jin, Yu
;
Wang, Shuo
;
Xu, Shujing
;
Zhao, Shujie
;
Xu, Xiangrui
, et al.
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Drug Discovery Today
July 2023 28(7)
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27 . Academic Journal
Discovery of novel sulfonamide substituted indolylarylsulfones as potent HIV-1 inhibitors with better safety profiles
저자
by
Gao, Shenghua
;
Song, Letian
;
Cheng, Yusen
;
Zhao, Fabao
;
Kang, Dongwei
, et al.
소스
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Acta Pharmaceutica Sinica B
June 2023 13(6):2747-2764
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27 . Academic Journal
Rapid discovery and crystallography study of highly potent and selective butylcholinesterase inhibitors based on oxime-containing libraries and conformational restriction strategies
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by
Jing, Lanlan
;
Wei, Wenxiu
;
Meng, Bairu
;
Chantegreil, Fabien
;
Nachon, Florian
, et al.
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Bioorganic Chemistry
May 2023 134
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27 . Academic Journal
Discovery of N-substituted oseltamivir derivatives as novel neuraminidase inhibitors with improved drug resistance profiles and favorable drug-like properties
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by
Jia, Ruifang
;
Zhang, Jiwei
;
Shi, Fangyuan
;
Bonomini, Anna
;
Lucca, Camilla
, et al.
소스
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European Journal of Medicinal Chemistry
5 April 2023 252
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27 . Academic Journal
Identification of “dual-site”-binding diarylpyrimidines targeting both NNIBP and the NNRTI adjacent site of the HIV-1 reverse transcriptase
저자
by
Feng, Da
;
Zuo, Xiaofang
;
Zhao, Fabao
;
Lin, Hao
;
Dai, Jiaojiao
, et al.
소스
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European Journal of Medicinal Chemistry
5 February 2023 247
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27 . Academic Journal
Disubstituted pyrimidine-5-carboxamide derivatives as novel HIV-1 NNRTIs: Crystallographic overlay-based molecular design, synthesis, and biological evaluation
저자
by
Feng, Da
;
Lin, Hao
;
Jiang, Liyang
;
Dai, Jiaojiao
;
Zhang, Xiaoying
, et al.
소스
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European Journal of Medicinal Chemistry
15 January 2023 246
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