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21 . Academic Journal
Discovery of Molecular Switches That Modulate Modes of Metabotropic Glutamate Receptor Subtype 5 (mGlu5) Pharmacology in Vitro and in Vivo within a Series of Functionalized, Regioisomeric 2- and 5-(Phenylethynyl)pyrimidines.
저자
by
Sameer Sharma
;
Jeffrey Kedrowski
;
Jerri M. Rook
;
Randy L. Smith
;
Carrie K. Jones
, et al.
소스
Journal of Medicinal Chemistry
. Jul2009, Vol. 52 Issue 14, p4103-4106. 4p.
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27 .
M 1 muscarinic activation induces long-lasting increase in intrinsic excitability of striatal projection neurons
저자
by
Zixiu Xiang
;
Jerri M. Rook
;
P. Jeffrey Conn
;
Jonathan W. Dickerson
;
Craig W. Lindsley
, et al.
소스
Neuropharmacology
. 118:209-222
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27 .
FUNCTIONAL ACTIVITY OF THE MUSCARINIC POSITIVE ALLOSTERIC MODULATOR VU319 DURING A PHASE 1 SINGLE ASCENDING DOSE STUDY
저자
by
Craig W. Lindsley
;
Jerri M. Rook
;
Paul A. Newhouse
;
Carrie K. Jones
;
Alexandra P. Key
, et al.
소스
The American Journal of Geriatric Psychiatry
. 28:S114-S115
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27 .
P4‐681: OPTIMIZATION OF NOVEL M1 PAMS FOR CLINICAL DEVELOPMENT WITH ENHANCED EFFICACY WHILE AVOIDING ADVERSE EFFECT LIABILITY FOR THE TREATMENT OF ALZHEIMER'S DISEASE
저자
by
Craig W. Lindsley
;
Jerri M. Rook
;
Paul A. Newhouse
;
P. Jeffrey Conn
.
소스
Alzheimer's & Dementia
. 15
Scopus
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26 .
Discovery of Tricyclic Triazolo- and Imidazopyridine Lactams as M(1) Positive Allosteric Modulators
저자
by
Jerri M. Rook
;
Colleen M. Niswender
;
Kyle A. Emmitte
;
Craig W. Lindsley
;
Jonathan W. Dickerson
, et al.
소스
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27 .
mGlu5positive allosteric modulation normalizes synaptic plasticity defects and motor phenotypes in a mouse model of Rett syndrome
저자
by
Jerri M. Rook
;
Rebecca K. Senter
;
Rocco G. Gogliotti
;
Shaun R. Stauffer
;
Carrie K. Jones
, et al.
소스
Human Molecular Genetics
. 25:1990-2004
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27 .
An mGlu5-Positive Allosteric Modulator Rescues the Neuroplasticity Deficits in a Genetic Model of NMDA Receptor Hypofunction in Schizophrenia
저자
by
Vadim Y. Bolshakov
;
Jerri M. Rook
;
Shunsuke Takagi
;
Darrick T. Balu
;
Carrie K. Jones
, et al.
소스
Neuropsychopharmacology
. 41:2052-2061
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27 .
Acyl dihydropyrazolo[1,5-a]pyrimidinones as metabotropic glutamate receptor 5 positive allosteric modulators
저자
by
José Manuel Bartolomé-Nebreda
;
Thomas Steckler
;
Susana Conde-Ceide
;
Colleen M. Niswender
;
Chrysa Malosh
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 25:5115-5120
Open Access (OpenAIRE)
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27 .
Development of Novel, CNS Penetrant Positive Allosteric Modulators for the Metabotropic Glutamate Receptor Subtype 1 (mGlu1), Based on an N-(3-Chloro-4-(1,3-dioxoisoindolin-2-yl)phenyl)-3-methylfuran-2-carboxamide Scaffold, That Potentiate Wild Type and Mutant mGlu1 Receptors Found in Schizophrenics
저자
by
Colleen M. Niswender
;
Hyekyung P. Cho
;
Jerri M. Rook
;
Anna L. Blobaum
;
P. Jeffrey Conn
, et al.
소스
Journal of Medicinal Chemistry
. 58:7959-7971
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27 .
Co-Activation of Metabotropic Glutamate Receptor 3 and Beta-Adrenergic Receptors Modulates Cyclic-AMP and Long-Term Potentiation, and Disrupts Memory Reconsolidation
저자
by
Adam G. Walker
;
Jerri M. Rook
;
Andrew S Lewis
;
Rebecca K. Senter
;
Douglas J. Sheffler
, et al.
소스
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