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21 .
Supplementary Methods from AZD9496: An Oral Estrogen Receptor Inhibitor That Blocks the Growth of ER-Positive and ESR1-Mutant Breast Tumors in Preclinical Models
저자
by
Chris De Savi
;
Celina D'Cruz
;
Anne Marie Mazzola
;
Ermira Pazolli
;
Brendon Ladd
, et al.
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27 .
Supplementary Figure 2 from Chromatin Remodeling Underlies the Senescence-Associated Secretory Phenotype of Tumor Stromal Fibroblasts That Supports Cancer Progression
저자
by
Sheila A. Stewart
;
David Piwnica-Worms
;
Julie Prior
;
Agnieszka Milczarek
;
Elise Alspach
, et al.
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27 .
Abstract P5-16-10: RLY-2608: The first allosteric mutant- and isoform-selective inhibitor of PI3Kα, is efficacious as a single agent and drives regressions in combination with standard of care therapies in PIK3CA mutant breast cancer models
저자
by
Ermira Pazolli
;
Randy Kipp
;
Alessandro Boezio
;
Hakan Gunaydin
;
Amanda Iskandar
, et al.
소스
Cancer Research
. 82:P5-16
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27 .
Sensitivity to splicing modulation of BCL2 family genes defines cancer therapeutic strategies for splicing modulators
저자
by
Zhenhua Jeremy Wu
;
Ermira Pazolli
;
Pete Smith
;
James Palacino
;
Deepti Banka
, et al.
소스
Nature Communications, Vol 10, Iss 1, Pp 1-15 (2019)
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27 .
Abstract P251: Discovery and characterization of RLY-2608: The first allosteric, mutant, and isoform-selective inhibitor of PI3Kα
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by
Ermira Pazolli
;
Randy Kipp
;
Alessandro Boezio
;
Hakan Gunaydin
;
Amanda Iskandar
, et al.
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Molecular Cancer Therapeutics
. 20:P251-P251
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27 .
Abstract DDT01-03: Discovery and pre-clinical pharmacology of AZD9496: An oral, selective estrogen receptor down-regulator (SERD)
저자
by
Anne Marie Mazzola
;
Graham Richmond
;
Craig S. Donald
;
Rachel Rowlinson
;
Celina M. D'Cruz
, et al.
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Cancer Research
. 75:DDT01-03
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27 .
c-Myb and C/EBPβ regulate OPN and other senescence-associated secretory phenotype factors
저자
by
Elise Alspach
;
Kevin C. Flanagan
;
Laura L. Arthur
;
Roberto Tapia
;
Ermira Pazolli
, et al.
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Oncotarget
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27 .
H3B-8800, an orally available small-molecule splicing modulator, induces lethality in spliceosome-mutant cancers
저자
by
Michael P. Thomas
;
Lihua Yu
;
Craig Karr
;
Eric Padron
;
Markus Warmuth
, et al.
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Nature medicine
. 24(4)
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27 .
p38MAPK Plays a Crucial Role in Stromal-Mediated Tumorigenesis
저자
by
Xianmin Luo
;
Sheila A. Stewart
;
Hui Huang
;
Megan K. Ruhland
;
Deborah V. Novack
, et al.
소스
Cancer Discovery
. 4:716-729
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27 .
Abstract 281: Sensitivity to splicing modulation of BCL2 family genes reveals cancer therapeutic strategies for splicing modulators
저자
by
Daniel Aird
;
Teng Teng
;
Chia-Ling Huang
;
Ermira Pazolli
;
Deepti Banka
, et al.
소스
Cancer Research
. 79:281-281
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