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11 . Academic Journal
Optimization of 1,2,4-Triazole-3-thiones toward Broad-Spectrum Metallo-β-lactamase Inhibitors Showing Potent Synergistic Activity on VIM- and NDM-1-Producing Clinical Isolates.
저자
by
Legru, Alice
;
Verdirosa, Federica
;
Vo-Hoang, Yen
;
Tassone, Giusy
;
Vascon, Filippo
, et al.
소스
Journal of Medicinal Chemistry; 12/22/2022, Vol. 65 Issue 24, p16392-16419, 28p
Full Text (ACS)
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17 . Academic Journal
Exploiting ELIOT for Scaffold-Repurposing Opportunities: TRIM33 a Possible Novel E3 Ligase to Expand the Toolbox for PROTAC Design.
저자
by
Palomba, Tommaso
;
Tassone, Giusy
;
Vacca, Carmine
;
Bartalucci, Matteo
;
Valeri, Aurora
, et al.
소스
International Journal of Molecular Sciences
. Nov2022, Vol. 23 Issue 22, p14218. 26p.
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17 . Academic Journal
Structural Basis of Parasitic HSP90 ATPase Inhibition by Small Molecules.
저자
by
Tassone, Giusy
;
Mazzorana, Marco
;
Pozzi, Cecilia
.
소스
Pharmaceuticals (14248247)
. Nov2022, Vol. 15 Issue 11, p1341. 21p.
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15 . Academic Journal
Mechanistic Aspects of the Asymmetric Transfer Hydrogenation in the Manufacture of Noradrenaline.
저자
by
Scorzelli, Francesco
;
Tassone, Giusy
;
Padula, Daniele
;
Zacchè, Matteo
.
소스
European Journal of Organic Chemistry
. 9/27/2022, Vol. 2022 Issue 36, p1-5. 5p.
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16 . Academic Journal
Structural Characterization of Human Heat Shock Protein 90 N-Terminal Domain and Its Variants K112R and K112A in Complex with a Potent 1,2,3-Triazole-Based Inhibitor.
저자
by
Tassone, Giusy
;
Mazzorana, Marco
;
Mangani, Stefano
;
Petricci, Elena
;
Cini, Elena
, et al.
소스
International Journal of Molecular Sciences
. Aug2022, Vol. 23 Issue 16, p9458-N.PAG. 11p.
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17 . Academic Journal
1,2,4‐Triazole‐3‐Thione Analogues with a 2‐Ethylbenzoic Acid at Position 4 as VIM‐type Metallo‐β‐Lactamase Inhibitors.
저자
by
Verdirosa, Federica
;
Gavara, Laurent
;
Sevaille, Laurent
;
Tassone, Giusy
;
Corsica, Giuseppina
, et al.
소스
ChemMedChem; 4/5/2022, Vol. 17 Issue 7, p1-13, 13p
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17 . Academic Journal
Xanthopsin‐Like Systems via Site‐Specific Click‐Functionalization of a Retinoic Acid Binding Protein.
저자
by
Tassone, Giusy
;
Paolino, Marco
;
Pozzi, Cecilia
;
Reale, Annalisa
;
Salvini, Laura
, et al.
소스
ChemBioChem; 1/5/2022, Vol. 23 Issue 1, p1-11, 11p
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17 . Academic Journal
Iron Binding in the Ferroxidase Site of Human Mitochondrial Ferritin.
저자
by
Ciambellotti, Silvia
;
Pratesi, Alessandro
;
Tassone, Giusy
;
Turano, Paola
;
Mangani, Stefano
, et al.
소스
Chemistry - A European Journal
. 10/21/2021, Vol. 27 Issue 59, p14690-14701. 12p.
Full Text (Wiley)
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17 . Academic Journal
Discovery of small molecule inhibitors of Leishmania braziliensis Hsp90 chaperone.
저자
by
Batista, Fernanda A. H.
;
Ramos, Sérgio L.
;
Tassone, Giusy
;
Leitão, Andrei
;
Montanari, Carlos A.
, et al.
소스
Journal of Enzyme Inhibition & Medicinal Chemistry
. Dec2020, Vol. 35 Issue 1, p639-649. 11p.
Open Access (T&F)
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17 . Academic Journal
High‐resolution crystal structure of Trypanosoma brucei pteridine reductase 1 in complex with an innovative tricyclic‐based inhibitor.
저자
by
Landi, Giacomo
;
Linciano, Pasquale
;
Tassone, Giusy
;
Costi, Maria Paola
;
Mangani, Stefano
, et al.
소스
Acta Crystallographica: Section D, Structural Biology
. Jun2020, Vol. 76 Issue 6, p558-564. 7p.
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