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11 . Academic Journal
The synthesis of tetrahydropyridopyrimidones as a new scaffold for HIV-1 integrase inhibitors
저자
by
Kinzel, Olaf D.
;
Monteagudo, Edith
;
Muraglia, Ester
;
Orvieto, Federica
;
Pescatore, Giovanna
, et al.
소스
Tetrahedron Letters: International Organ for the Rapid Publication of Preliminary Communications in Organic Chemistry
. Sep2007, Vol. 48 Issue 37, p6552-6555. 4p.
Full Text (ScienceDirect)
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17 . Academic Journal
Polypharmacy through Phage Display: Selection of Glucagon and GLP-1 Receptor Co-agonists from a Phage-Displayed Peptide Library
저자
by
Demartis, Anna
;
Lahm, Armin
;
Tomei, Licia
;
Beghetto, Elisa
;
Di Biasio, Valentina
, et al.
소스
SCIENTIFIC REPORTS
; JAN 12 2018, 8 p585 9p.
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17 . Academic Journal
An Expedient Synthesis of 14,14-Dimethyl-3,7-diazatricyclo[8.3.1 .0 ]tetradec-7-en-4-one-12α-yl Cinnamate, an Unusual Heterocyclic Compound Resembling the A/B/C Core of Taxanes.
저자
by
Orvieto, Federica
;
Botta, Maurizio
;
Corelli, Federico
;
Harper, Steven
.
소스
Synthetic Communications; Oct1999, Vol. 29 Issue 20, p3635-3649, 15p
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16 . Patent
저자
by
Merck Sharp & Dohme Corp.
;
Palani, Anandan
;
Nargund, Ravi
;
Carrington, Paul E.
;
Sawyer, Tomi
, et al.
소스
Open Access (USPTO)
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17 . Periodical
An Expedient Synthesis of 14,14-Dimethyl-3,7-diazatricyclo[8.3.11,10.03.8]tetradec-7-en-4-one-12α-yl Cinnamate, an Unusual Heterocyclic Compound Resembling the A/B/C Core of Taxanes
저자
by
Orvieto, Federica
;
Botta, Maurizio
;
Corelli, Federico
;
Harper, Steven
.
소스
Synthetic Communications; October 1999, Vol. 29 Issue: 20 p3635-3649, 15p
Web of Science
Scopus
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16 . Academic Journal
Discovery of Raltegravir, a potent, selective orally bioavailable HIV-integrase inhibitor for the treatment of HIV-AIDS infection
저자
by
Summa, Vincenzo
;
Petrocchi, Alessia
;
Bonelli, Fabio
;
Crescenzi, Benedetta
;
Donghi, Monica
, et al.
소스
JOURNAL OF MEDICINAL CHEMISTRY
; SEP 25 2008, 51 18, p5843-p5855, 13p.
Full Text (ACS)
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17 . Academic Journal
Design and synthesis of bicyclic pyrimidinones as potent and orally bioavailable HIV-1 integrase inhibitors
저자
by
Muraglia, Ester
;
Kinzel, Olaf
;
Gardelli, Cristina
;
Crescenzi, Benedetta
;
Donghi, Monica
, et al.
소스
JOURNAL OF MEDICINAL CHEMISTRY
; FEB 28 2008, 51 4, p861-p874, 14p.
Full Text (ACS)
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17 . Academic Journal
Discovery and synthesis of HIV integrase inhibitors: Development of potent and orally bioavailable N-methyl Pyrimidones
저자
by
Gardelli, Cristina
;
Nizi, Emanuela
;
Muraglia, Ester
;
Crescenzi, Benedetta
;
Ferrara, Marco
, et al.
소스
JOURNAL OF MEDICINAL CHEMISTRY
; OCT 4 2007, 50 20, p4953-p4975, 23p.
Full Text (ACS)
Scopus
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17 . Academic Journal
Dihydroxypyrimidine-4-carboxamides as novel potent and selective HIV integrase inhibitors
저자
by
Pace, Paola
;
Di Francesco, M. Emilia
;
Gardelli, Cristina
;
Harper, Steven
;
Muraglia, Ester
, et al.
소스
JOURNAL OF MEDICINAL CHEMISTRY
; MAY 3 2007, 50 9, p2225-p2239, 15p.
Full Text (ACS)
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17 . Patent
저자
by
Boueres, Julia
;
Branca, Danila
;
Ferrigno, Federica
;
Jones, Philip
;
Muraglia, Ester
, et al.
소스
Open Access (USPTO)
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