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11 . Academic Journal
Discovery of TRPM8 Antagonist (S)‑6-(((3-Fluoro-4-(trifluoromethoxy)phenyl)(3-fluoropyridin-2-yl)methyl)carbamoyl)nicotinic Acid (AMG 333), a Clinical Candidate for the Treatment of Migraine.
저자
by
Horne, Daniel B.
;
Biswas, Kaustav
;
Brown, James
;
Bartberger, Michael D.
;
Clarine, Jeffrey
, et al.
소스
Journal of Medicinal Chemistry; 9/27/2018, Vol. 61 Issue 18, p8186-8201, 16p
Full Text (ACS)
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17 . Academic Journal
Development of TRPM8 Antagonists to Treat Chronic Pain and Migraine.
저자
by
Weyer, Andy D.
;
Lehto, Sonya G.
.
소스
Pharmaceuticals (14248247)
. Jun2017, Vol. 10 Issue 2, p37. 9p.
Web of Science
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14 . Academic Journal
The Discovery and Hit-to-Lead Optimization of Tricyclic Sulfonamides as Potent and Efficacious Potentiators of Glycine Receptors.
저자
by
Bregman, Howard
;
Simard, Jeffrey R.
;
Andrews, Kristin L.
;
Ayube, Shawn
;
Hao Chen
, et al.
소스
Journal of Medicinal Chemistry
. Feb2017, Vol. 60 Issue 3, p1105-1125. 21p.
Full Text (ACS)
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17 . Academic Journal
Optimization of a Novel Quinazolinone-Based Series of Transient Receptor Potential A1 (TRPA1) Antagonists Demonstrating Potent in Vivo Activity.
저자
by
Schenkel, Laurie B.
;
Olivieri, Philip R.
;
Boezio, Alessandro A.
;
Deak, Holly L.
;
Emkey, Renee
, et al.
소스
Journal of Medicinal Chemistry
. Mar2016, Vol. 59 Issue 6, p2794-2809. 16p.
Full Text (ACS)
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17 . Academic Journal
Voltage-gated sodium channel function and expression in injured and uninjured rat dorsal root ganglia neurons.
저자
by
Yin, Ruoyuan
;
Liu, Dong
;
Chhoa, Mark
;
Li, Chi-Ming
;
Luo, Yi
, et al.
소스
International Journal of Neuroscience
. Feb2016, Vol. 126 Issue 2, p182-192. 11p.
Web of Science
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17 . Academic Journal
Selective antagonism of TRPA1 produces limited efficacy in models of inflammatoryand neuropathic-induced mechanical hypersensitivity in rats.
저자
by
Lehto, Sonya G.
;
Weyer, Andy D.
;
Youngblood, Beth D.
;
Maosheng Zhang
;
Ruoyuan Yin
, et al.
소스
Molecular Pain
. 2016, Vol. 12, p1-13. 13p. 2 Charts, 4 Graphs.
Full Text (Sage OA)
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17 . Academic Journal
Optimization of Potency andPharmacokinetic Propertiesof Tetrahydroisoquinoline Transient Receptor Potential Melastatin8 (TRPM8) Antagonists.
저자
by
Horne, Daniel B.
;
Tamayo, Nuria A.
;
Bartberger, Michael D.
;
Bo, Yunxin
;
Clarine, Jeffrey
, et al.
소스
Journal of Medicinal Chemistry
. Apr2014, Vol. 57 Issue 7, p2989-3004. 16p.
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17 . Academic Journal
Transient Receptor Potential Channel Ankyrin-1 Is Not a Cold Sensor for Autonomic Thermoregulation in Rodents.
저자
by
de Oliveira, Cristiane
;
Garami, Andras
;
Lehto, Sonya G.
;
Pakai, Eszter
;
Tekus, Valeria
, et al.
소스
Journal of Neuroscience
. 3/26/2014, Vol. 34 Issue 13, p4445-4452. 8p.
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17 . Academic Journal
Fused Piperidines as aNovel Class of Potent and OrallyAvailable Transient Receptor Potential Melastatin Type 8 (TRPM8) Antagonists.
저자
by
Tamayo, Nuria A.
;
Bo, Yunxin
;
Gore, Vijay
;
Ma, Vu
;
Nishimura, Nobuko
, et al.
소스
Journal of Medicinal Chemistry
. Feb2012, Vol. 55 Issue 4, p1593-1611. 19p.
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17 . Academic Journal
Transient receptor potential melastatin 8 (TRPM8) channels are involved in body temperature regulation.
저자
by
Gavva, Narender R.
;
Davis, Carl
;
Lehto, Sonya G.
;
Rao, Sara
;
Wang, Weiya
, et al.
소스
Molecular Pain
. 2012, Vol. 8 Issue 1, p36-44. 9p. 3 Diagrams, 2 Charts.
Open Access (BioMed Central)
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