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11 .
539. GS-CA2: A Novel, Potent, and Selective First-In-class Inhibitor of HIV-1 Capsid Function Displays Nonclinical Pharmacokinetics Supporting Long-Acting Potential in Humans
저자
by
Schroeder Scott D
;
Tse Winston C
;
Raju Subramanian
;
Anna Chiu
;
Tomas Cihlar
, et al.
소스
Open Forum Infectious Diseases
Open Access (OpenAIRE)
Web of Science
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17 .
Abyssomicin 2 Reactivates Latent HIV-1 by a PKC- and HDAC-Independent Mechanism
저자
by
Angela Tsai
;
George Stepan
;
Nikos Pagratis
;
Gregg S. Jones
;
Bailey J Dickey
, et al.
소스
Organic Letters
. 17:262-265
Open Access (OpenAIRE)
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17 .
Study of Marine Natural Products Including Resorcyclic Acid Lactones from Humicola fuscoatra That Reactivate Latent HIV-1 Expression in an in Vitro Model of Central Memory CD4+ T Cells
저자
by
Tomas Cihlar
;
Tiffany Barnes
;
Karen Tenney
;
Eric J. Mejia
;
Romas Geleziunas
, et al.
소스
Journal of Natural Products
Open Access (OpenAIRE)
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17 .
Novel (2,6-difluorophenyl)(2-(phenylamino)pyrimidin-4-yl)methanones with restricted conformation as potent non-nucleoside reverse transcriptase inhibitors against HIV-1
저자
by
George Stepan
;
Ondřej Baszczyňski
;
Eric B. Lansdon
;
Petr Šimon
;
David Šaman
, et al.
소스
European journal of medicinal chemistry
. 122
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17 .
Effect of YM-44781, YM-44778 and YM-49598, Novel Tachykinin Antagonists, in a Drug-Induced Bladder Contraction Model
저자
by
Gretchen Groke
;
Analyn Bringas
;
Michael Patrick Dillon
;
George Stepan
;
A. Choppin
.
소스
Pharmacology
. 65:96-102
Web of Science
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17 .
Inhibition of hepatitis C virus replication by GS-6620, a potent C-nucleoside monophosphate prodrug
저자
by
Betty Peng
;
Yang Tian
;
Choung U. Kim
;
Joy Y. Feng
;
Aesop Cho
, et al.
소스
Antimicrobial agents and chemotherapy
. 58(4)
Full Text (ASM)
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17 .
9-[2-(R)-(Phosphonomethoxy)propyl]-2,6-diaminopurine (R)-PMPDAP and its prodrugs: optimized preparation, including identification of by-products formed, and antiviral evaluation in vitro
저자
by
Joeri Auwerx
;
Václav Kašička
;
Eleonora Kiss
;
George Stepan
;
Petr Jansa
, et al.
소스
Bioorganic & Medicinal Chemistry
Full Text (ScienceDirect)
Open Access (OpenAIRE)
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17 .
Search for small molecule activators of latent HIV
저자
by
Joe Hesselgesser
;
Nikos Pagratis
;
Helen Yu
;
George Wei
;
Romas Geleziunas
, et al.
소스
Retrovirology, Vol 9, Iss Suppl 1, p O2 (2012)
Retrovirology
Open Access (BioMed Central)
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17 .
Histone Deacetylase Inhibitor Romidepsin Induces HIV Expression in CD4 T Cells from Patients on Suppressive Antiretroviral Therapy at Concentrations Achieved by Clinical Dosing
저자
by
Joseph Hesselgesser
;
Alivelu Irrinki
;
Jacob Lalezari
;
Vicki Chiang
;
Mini Balakrishnan
, et al.
소스
PLoS Pathogens
PLoS Pathogens, Vol 10, Iss 4, p e1004071 (2014)
Open Access (OpenAIRE)
Web of Science
Scopus
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17 .
Human cloned alpha1A-adrenoceptor isoforms display alpha1L-adrenoceptor pharmacology in functional studies
저자
by
David J. Chang
;
John D Lesnick
;
Jeffrey R. Jasper
;
David E. Clarke
;
Donald V. Daniels
, et al.
소스
European journal of pharmacology
. 370(3)
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