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11 .
Analysis by substituted cysteine scanning mutagenesis of the fourth transmembrane domain of the CXCR4 receptor in its inactive and active state
저자
by
Philip E. Boulais
;
Richard Leduc
;
Emanuel Escher
.
소스
Biochemical Pharmacology
. 85:541-550
Web of Science
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15 .
Structure-Activity Relationship and Signaling of New Chimeric CXCR4 Agonists
저자
by
Nikolaus Heveker
;
Jérôme Cabana
;
Marilou Lefrançois
;
Marie-Reine Lefebvre
;
Christine E. Mona
, et al.
소스
Journal of medicinal chemistry
. 59(16)
Scopus
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17 .
Identification of Membrane-bound Variant of Metalloendopeptidase Neurolysin (EC 3.4.24.16) as the Non-angiotensin Type 1 (Non-AT1), Non-AT2 Angiotensin Binding Site
저자
by
Kira L. Santos
;
Fred K. Hagen
;
Robert C. Speth
;
Vardan T. Karamyan
;
Emanuel Escher
, et al.
소스
Journal of Biological Chemistry
. 287:114-122
Open Access (OpenAIRE)
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17 .
Angiotensin II Analogues with Sulphur-containing Side-chains in Position 5
저자
by
Vassiliki Magafa
;
Richard Bouley
;
Emanuel Escher
;
Jacqueline Pérodin
;
Dimitrios Theodoropoulos
, et al.
소스
Arzneimittelforschung
. 50:526-529
Scopus
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17 .
A single-nucleotide polymorphism of alanine to threonine at position 163 of the human angiotensin II type 1 receptor impairs Losartan affinity
저자
by
Jason Arsenault
;
Gaétan Guillemette
;
Jérôme Cabana
;
Pierre Lavigne
;
Emanuel Escher
, et al.
소스
Pharmacogenetics and Genomics
. 20:377-388
Full Text (LWW)
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17 .
Preliminary biochemical characterization of the novel, non-AT1, non-AT2 angiotensin binding site from the rat brain
저자
by
Robert C. Speth
;
Vardan T. Karamyan
;
Jason Arsenault
;
Emanuel Escher
.
소스
Endocrine
. 37:442-448
Open Access (OpenAIRE)
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16 .
The Amino-Terminus of Angiotensin II Contacts Several Ectodomains of the Angiotensin II Receptor AT1
저자
by
Gaétan Guillemette
;
Luta Luse Basambombo
;
Richard Leduc
;
Guillaume Lemieux
;
Dany Fillion
, et al.
소스
Journal of Medicinal Chemistry
. 53:2063-2075
Web of Science
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17 .
Analysis of Transmembrane Domains 1 and 4 of the Human Angiotensin II AT1 Receptor by Cysteine-scanning Mutagenesis
저자
by
Richard Leduc
;
Gaétan Guillemette
;
Brian J. Holleran
;
Emanuel Escher
;
Liping Yan
, et al.
소스
Journal of Biological Chemistry
. 285:2284-2293
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17 .
The Second Transmembrane Domain of the Human Type 1 Angiotensin II Receptor Participates in the Formation of the Ligand Binding Pocket and Undergoes Integral Pivoting Movement during the Process of Receptor Activation
저자
by
Ivana Domazet
;
Brian J. Holleran
;
Richard Leduc
;
Emanuel Escher
;
Pierre Lavigne
, et al.
소스
Journal of Biological Chemistry
. 284:11922-11929
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17 .
Synthesis of new head-activator analogues and their application for improved radioimmunoassays
저자
by
H. Bodenmüller
;
E. Schilling
;
Emanuel Escher
;
B. Zachmann
.
소스
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