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1 . Academic Journal
NIBR-LTSi is a selective LATS kinase inhibitor activating YAP signaling and expanding tissue stem cells in vitro and in vivo
저자
by
Namoto, Kenji
;
Baader, Clara
;
Orsini, Vanessa
;
Landshammer, Alexandro
;
Breuer, Eva
, et al.
소스
In
Cell Stem Cell
4 April 2024 31(4):554-569
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7 . Academic Journal
Small-molecule factor B inhibitor for the treatment of complement-mediated diseases
저자
by
Schubart, Anna
;
Anderson, Karen
;
Mainolfi, Nello
;
Sellner, Holger
;
Ehara, Takeru
, et al.
소스
Proceedings of the National Academy of Sciences of the United States of America, 2019 Apr . 116(16), 7926-7931.
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7 .
Small-molecule factor D inhibitors targeting the alternative complement pathway
저자
by
Frederic Cumin
;
Bernd Kinzel
;
Anna Vulpetti
;
Antonio M. Risitano
;
Richard A. Harrison
, et al.
소스
Nature chemical biology
. 12(12)
Open Access (OpenAIRE)
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7 .
Discovery of 4-((2S,4S)-4-Ethoxy-1-((5-methoxy-7-methyl-1H-indol-4-yl)methyl)piperidin-2-yl)benzoic Acid (LNP023), a Factor B Inhibitor Specifically Designed To Be Applicable to Treating a Diverse Array of Complement Mediated Diseases
저자
by
Nello Mainolfi
;
Takeru Ehara
;
Rajeshri G. Karki
;
Karen Anderson
;
Aengus Mac Sweeney
, et al.
소스
Journal of Medicinal Chemistry
. 63:5697-5722
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7 .
Discovery and Design of First Benzylamine-Based Ligands Binding to an Unlocked Conformation of the Complement Factor D
저자
by
A. Mac Sweeney
;
Jürgen Maibaum
;
Edwige Liliane Jeanne Lorthiois
;
Simon Rüdisser
;
Frederic Cumin
, et al.
소스
ACS Medicinal Chemistry Letters
. 9:490-495
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7 .
Discovery of Highly Potent and Selective Small-Molecule Reversible Factor D Inhibitors Demonstrating Alternative Complement Pathway Inhibition in Vivo
저자
by
Stefanie Flohr
;
Simon Rüdisser
;
Anna Vulpetti
;
Andrea De Erkenez
;
Stefan Steinbacher
, et al.
소스
Journal of Medicinal Chemistry
. 60:5717-5735
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7 .
Structure-Based Library Design and Fragment Screening for the Identification of Reversible Complement Factor D Protease Inhibitors
저자
by
Paul Erbel
;
Bernd Gerhartz
;
Frederic Cumin
;
Jürgen Maibaum
;
Nils Ostermann
, et al.
소스
Journal of Medicinal Chemistry
. 60:1946-1958
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7 .
trans -(3 S ,4 S )-Disubstituted pyrrolidines as inhibitors of the human aspartyl protease renin. Part I: Prime site exploration using an amino linker
저자
by
Claus Ehrhardt
;
Jürgen Maibaum
;
Edwige Lorthiois
;
Takatoshi Kosaka
;
Nils Ostermann
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 25:1782-1786
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7 .
Structure-Based Design of Substituted Piperidines as a New Class of Highly Efficacious Oral Direct Renin Inhibitors
저자
by
Shimpei Kawakami
;
Nikolaus Schiering
;
Takeru Ehara
;
Fumiaki Yokokawa
;
Hiroki Gunji
, et al.
소스
ACS Medicinal Chemistry Letters
. 5:787-792
Open Access (OpenAIRE)
Web of Science
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7 . Academic Journal
Discovery and Design of First Benzylamine-Based Ligands Binding to an Unlocked Conformation of the Complement Factor D
저자
by
Vulpetti, Anna
;
Ostermann, Nils
;
Randl, Stefan
;
Yoon, Taeyoung
;
Mac Sweeney, Aengus
, et al.
소스
ACS MEDICINAL CHEMISTRY LETTERS
; MAY 2018, 9 5, p490-p495, 11p.
Full Text (ACS)
Scopus
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