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1 . Academic Journal
Discovery of novel multifunctional ligands targeting GABA transporters, butyrylcholinesterase, β-secretase, and amyloid β aggregation as potential treatment of Alzheimer's disease
저자
by
Zaręba, Paula
;
Łątka, Kamil
;
Mazur, Gabriela
;
Gryzło, Beata
;
Pasieka, Anna
, et al.
소스
In
European Journal of Medicinal Chemistry
5 December 2023 261
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7 . Academic Journal
Development of tricyclic N-benzyl-4-hydroxybutanamide derivatives as inhibitors of GABA transporters mGAT1-4 with anticonvulsant, antinociceptive, and antidepressant activity
저자
by
Zaręba, Paula
;
Sałat, Kinga
;
Höfner, Georg C.
;
Łątka, Kamil
;
Bajda, Marek
, et al.
소스
In
European Journal of Medicinal Chemistry
5 October 2021 221
Full Text (ScienceDirect)
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7 . Academic Journal
Novel mouse GABA uptake inhibitors with enhanced inhibitory activity toward mGAT3/4 and their effect on pain threshold in mice
저자
by
Zaręba, Paula
;
Gryzło, Beata
;
Malawska, Katarzyna
;
Sałat, Kinga
;
Höfner, Georg C.
, et al.
소스
In
European Journal of Medicinal Chemistry
15 February 2020 188
Full Text (ScienceDirect)
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7 . Academic Journal
Development, validation and application of a 96-well enzymatic assay based on LC-ESI-MS/MS quantification for the screening of selective inhibitors against Mycobacterium tuberculosis purine nucleoside phosphorylase
저자
by
Cattaneo, Giulia
;
Ubiali, Daniela
;
Calleri, Enrica
;
Rabuffetti, Marco
;
Höfner, Georg C.
, et al.
소스
In
Analytica Chimica Acta
2 November 2016 943:89-97
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7 .
Determination of enantiomeric excess of nipecotic acid as 1-(7-nitrobenzo[
c
][1,2,5]oxadiazol-4-yl) derivatives
저자
by
Simone K. Schmidt
;
Georg Höfner
;
Klaus T. Wanner
.
소스
Chirality
. 29:48-56
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5 . Academic Journal
Synthesis, biological evaluation and structure–activity relationship of new GABA uptake inhibitors, derivatives of 4-aminobutanamides
저자
by
Kowalczyk, Paula
;
Sałat, Kinga
;
Höfner, Georg C.
;
Mucha, Marta
;
Rapacz, Anna
, et al.
소스
In
European Journal of Medicinal Chemistry
18 August 2014 83:256-273
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7 . Academic Journal
2-Substituted 4-hydroxybutanamides as potential inhibitors of γ-aminobutyric acid transporters mGAT1–mGAT4: Synthesis and biological evaluation
저자
by
Kowalczyk, Paula
;
Sałat, Kinga
;
Höfner, Georg C.
;
Guzior, Natalia
;
Filipek, Barbara
, et al.
소스
In
Bioorganic & Medicinal Chemistry
1 September 2013 21(17):5154-5167
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7 . Academic Journal
Synthesis and biological evaluation of 4-hydroxy-4-(4-methoxyphenyl)-substituted proline and pyrrolidin-2-ylacetic acid derivatives as GABA uptake inhibitors
저자
by
Zhao, Xueqing
;
Pabel, Jörg
;
Höfner, Georg C.
;
Wanner, Klaus T.
.
소스
In
Bioorganic & Medicinal Chemistry
15 January 2013 21(2):470-484
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6 . Academic Journal
Azidobupramine, an Antidepressant-Derived Bifunctional Neurotransmitter Transporter Ligand Allowing Covalent Labeling and Attachment of Fluorophores.
저자
by
Thomas Kirmeier
;
Ranganath Gopalakrishnan
;
Vanessa Gormanns
;
Anna M Werner
;
Serena Cuboni
, et al.
소스
PLoS ONE, Vol 11, Iss 2, p e0148608 (2016)
Open Access (DOAJ)
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7 .
Synthesis and biological evaluation of α- and β-hydroxy substituted amino acid derivatives as potential mGAT1–4 inhibitors
저자
by
Georg Höfner
;
Michael C. Böck
;
Klaus T. Wanner
;
Janina C. Andreß
.
소스
Medicinal Chemistry Research
. 29:1321-1340
Open Access (OpenAIRE)
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