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1 . Academic Journal
Development of potential preclinical candidates with promising in vitro ADME profile for the inhibition of type 1 and type 2 17β-Hydroxysteroid dehydrogenases: Design, synthesis, and biological evaluation
저자
by
Abdelsamie, Ahmed S.
;
Salah, Mohamed
;
Siebenbürger, Lorenz
;
Hamed, Mostafa M.
;
Börger, Carsten
, et al.
소스
In
European Journal of Medicinal Chemistry
15 September 2019 178:93-107
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7 . Academic Journal
Treatment of estrogen-dependent diseases: Design, synthesis and profiling of a selective 17β-HSD1 inhibitor with sub-nanomolar IC50 for a proof-of-principle study
저자
by
Abdelsamie, Ahmed S.
;
van Koppen, Chris J.
;
Bey, Emmanuel
;
Salah, Mohamed
;
Börger, Carsten
, et al.
소스
In
European Journal of Medicinal Chemistry
15 February 2017 127:944-957
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7 . Academic Journal
Towards the evaluation in an animal disease model: Fluorinated 17β-HSD1 inhibitors showing strong activity towards both the human and the rat enzyme
저자
by
Abdelsamie, Ahmed S.
;
Bey, Emmanuel
;
Gargano, Emanuele M.
;
van Koppen, Chris J.
;
Empting, Martin
, et al.
소스
In
European Journal of Medicinal Chemistry
20 October 2015 103:56-68
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7 . Academic Journal
Potent Dual Inhibitors of Steroid Sulfatase and 17β-Hydroxysteroid Dehydrogenase Type 1 with a Suitable Pharmacokinetic Profile for In Vivo Proof-of-Principle Studies in an Endometriosis Mouse Model.
저자
by
Salah, Mohamed
;
Tahoun, Mariam
;
Rudzitis-Auth, Jeannette
;
Stotz, Lisa
;
van Koppen, Chris J.
, et al.
소스
Journal of Medicinal Chemistry; 7/13/2023, Vol. 66 Issue 13, p8975-8992, 18p
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7 . Academic Journal
Pharmacological Characterization of Receptor Redistribution and β-Arrestin Recruitment Assays for the Cannabinoid Receptor 1
저자
by
Van Der Lee, Miranda M.C.
;
Blomenröhr, Marion
;
Van Der Doelen, Antoon A.
;
Wat, Jesse W.Y.
;
Smits, Niels
, et al.
소스
In
SLAS Discovery
August 2009 14(7):811-823
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7 . Academic Journal
β-Arrestin Recruitment Assay for the Identification of Agonists of the Sphingosine 1-Phosphate Receptor EDG1
저자
by
Van Der Lee, Miranda M.C.
;
Bras, Maaike
;
Van Koppen, Chris J.
;
Zaman, Guido J.R.
.
소스
In
SLAS Discovery
December 2008 13(10):986-998
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6 . Academic Journal
Cryopreserved cells facilitate cell-based drug discovery
저자
by
Zaman, Guido J.R.
;
de Roos, Jeroen A.D.M.
;
Blomenröhr, Marion
;
van Koppen, Chris J.
;
Oosterom, Julia
.
소스
In
Drug Discovery Today
2007 12(13):521-526
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7 . Academic Journal
Accelerated skin wound healing by selective 11β-Hydroxylase (CYP11B1) inhibitors
저자
by
Emmerich, Juliette
;
van Koppen, Chris J.
;
Burkhart, Jens L.
;
Engeli, Roger T.
;
Hu, Qingzhong
, et al.
소스
In
European Journal of Medicinal Chemistry
1 January 2018 143:591-597
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7 . Academic Journal
Muscarinic receptors in the Mammalian Heart
저자
by
Dhein, Stefan
;
van Koppen, Chris J.
;
Brodde, Otto-Erich
.
소스
In
Pharmacological Research
September 2001 44(3):161-182
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5 . Academic Journal
17β-Hydroxysteroid Dehydrogenase Type 1 Inhibition: A Potential Treatment Option for Non-Small Cell Lung Cancer.
저자
by
Gargano, Emanuele M.
;
Mohamed, Abdelrahman
;
Abdelsamie, Ahmed S.
;
Mangiatordi, Giuseppe F.
;
Drzewiecka, Hanna
, et al.
소스
ACS Medicinal Chemistry Letters; 12/9/2021, Vol. 12 Issue 12, p1920-1924, 5p
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