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1 . Academic Journal
Novel 6-alkyl-bridged 4-arylalkylpiperazin-1-yl derivatives of azepino[4,3-b]indol-1(2H)-one as potent BChE-selective inhibitors showing protective effects against neurodegenerative insults
저자
by
Samarelli, Francesco
;
Purgatorio, Rosa
;
Lopopolo, Gianfranco
;
Deruvo, Caterina
;
Catto, Marco
, et al.
소스
In
European Journal of Medicinal Chemistry
15 April 2024 270
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7 . Academic Journal
A second life for MAO inhibitors? From CNS diseases to anticancer therapy
저자
by
Sblano, Sabina
;
Boccarelli, Angelina
;
Mesiti, Francesco
;
Purgatorio, Rosa
;
de Candia, Modesto
, et al.
소스
In
European Journal of Medicinal Chemistry
5 March 2024 267
Full Text (ScienceDirect)
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7 . Academic Journal
In-vitro and in-silico studies of annelated 1,4,7,8-tetrahydroazocine ester derivatives as nanomolar selective inhibitors of human butyrylcholinesterase
저자
by
de Candia, Modesto
;
Titov, Alexander A.
;
Viayna, Antonio
;
Kulikova, Larisa N.
;
Purgatorio, Rosa
, et al.
소스
In
Chemico-Biological Interactions
1 December 2023 386
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7 . Academic Journal
Synthesis, computational and experimental pharmacological studies for (thio)ether-triazine 5-HT6R ligands with noticeable action on AChE/BChE and chalcogen-dependent intrinsic activity in search for new class of drugs against Alzheimer's disease
저자
by
Czarnota-Łydka, Kinga
;
Sudoł-Tałaj, Sylwia
;
Kucwaj-Brysz, Katarzyna
;
Kurczab, Rafał
;
Satała, Grzegorz
, et al.
소스
In
European Journal of Medicinal Chemistry
5 November 2023 259
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7 . Academic Journal
Investigating 1,2,3,4,5,6-hexahydroazepino[4,3-b]indole as scaffold of butyrylcholinesterase-selective inhibitors with additional neuroprotective activities for Alzheimer's disease
저자
by
Purgatorio, Rosa
;
de Candia, Modesto
;
Catto, Marco
;
Carrieri, Antonio
;
Pisani, Leonardo
, et al.
소스
In
European Journal of Medicinal Chemistry
1 September 2019 177:414-424
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7 . Academic Journal
Nature-Inspired 1-Phenylpyrrolo[2,1- a ]isoquinoline Scaffold for Novel Antiproliferative Agents Circumventing P-Glycoprotein-Dependent Multidrug Resistance.
저자
by
Nevskaya, Alisa A.
;
Purgatorio, Rosa
;
Borisova, Tatiana N.
;
Varlamov, Alexey V.
;
Anikina, Lada V.
, et al.
소스
Pharmaceuticals (14248247)
. Apr2024, Vol. 17 Issue 4, p539. 17p.
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7 . Academic Journal
Targeting a Mirabegron precursor by BH3-mediated continuous flow reduction process
저자
by
De Angelis, Sonia
;
Carlucci, Claudia
;
de Candia, Modesto
;
Rebuzzini, Gabriele
;
Celestini, Paolo
, et al.
소스
In
Catalysis Today
15 June 2018 308:81-85
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7 . Academic Journal
The position of fluorine in CP-118,954 affects AChE inhibition potency and PET imaging quantification for AChE expression in the rat brain
저자
by
Lee, Byung Chul
;
Moon, Byung Seok
;
Park, Hyun Soo
;
Jung, Jae Ho
;
Park, Hyun Sik
, et al.
소스
In
European Journal of Pharmaceutical Sciences
15 November 2017 109:209-216
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7 . Academic Journal
Pharmaceutical development of novel lactate-based 6-fluoro-l-DOPA formulations
저자
by
Denora, Nunzio
;
Lopedota, Angela
;
de Candia, Modesto
;
Cellamare, Saverio
;
Degennaro, Leonardo
, et al.
소스
In
European Journal of Pharmaceutical Sciences
1 March 2017 99:361-368
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7 . Academic Journal
New azepino[4,3-b]indole derivatives as nanomolar selective inhibitors of human butyrylcholinesterase showing protective effects against NMDA-induced neurotoxicity
저자
by
de Candia, Modesto
;
Zaetta, Giorgia
;
Denora, Nunzio
;
Tricarico, Domenico
;
Majellaro, Maria
, et al.
소스
In
European Journal of Medicinal Chemistry
5 January 2017 125:288-298
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