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1 . Academic Journal
Discovery and Characterization of Potent, Efficacious, Orally Available Antimalarial Plasmepsin X Inhibitors and Preclinical Safety Assessment of UCB7362.
저자
by
Lowe, Martin A.
;
Cardenas, Alvaro
;
Valentin, Jean-Pierre
;
Zhu, Zhaoning
;
Abendroth, Jan
, et al.
소스
Journal of Medicinal Chemistry; 10/27/2022, Vol. 65 Issue 20, p14121-14143, 23p
Full Text (ACS)
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7 . Academic Journal
Discovery of potent iminoheterocycle BACE1 inhibitors
저자
by
Caldwell, John P.
;
Mazzola, Robert D.
;
Durkin, James
;
Chen, Joseph
;
Chen, Xia
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 December 2014 24(23):5455-5459
Full Text (ScienceDirect)
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7 . Academic Journal
Unprecedented Reversal of Regioselectivity during Methanolysis and an Interception of Curtius Rearrangement.
저자
by
Mandal, Mihirbaran
;
Buevich, Alexei V.
;
Wang, Hongwu
;
Brunskill, Andrew
;
Orth, Peter
, et al.
소스
European Journal of Organic Chemistry
. 9/24/2021, Vol. 2021 Issue 36, p5073-5079. 7p.
Web of Science
Scopus
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7 . Academic Journal
The discovery of fused oxadiazepines as gamma secretase modulators for treatment of Alzheimer’s disease
저자
by
Li, Hongmei
;
Qin, Jun
;
Dhondi, Pawan
;
Zhou, Wei
;
Vicarel, Monica
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 January 2013 23(2):466-471
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7 . Academic Journal
On the power of super acid—iodination of aromatic ring in the presence of imidazole moiety of the potent gamma secretase modulators (GSM) en route to tritium labeling
저자
by
Mandal, Mihirbaran
;
Lavey, Carolee
;
Buevich, Alexei V.
;
Zhu, Zhaoning
;
Stamford, Andrew W.
, et al.
소스
In
Tetrahedron Letters
4 April 2012 53(14):1725-1727
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7 . Academic Journal
Structure based design of iminohydantoin BACE1 inhibitors: Identification of an orally available, centrally active BACE1 inhibitor
저자
by
Cumming, Jared N.
;
Smith, Elizabeth M.
;
Wang, Lingyan
;
Misiaszek, Jeffrey
;
Durkin, James
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 April 2012 22(7):2444-2449
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7 . Academic Journal
Generation of Leads for γ‑Secretase Modulation.
저자
by
Mandal, Mihirbaran
;
Buevich, Alexei
;
Caldwell, John P.
;
Hyde, Lynn
;
Huang, Xianhai
, et al.
소스
Journal of Medicinal Chemistry; 8/13/2020, Vol. 63 Issue 15, p8216-8230, 15p
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7 . Academic Journal
Discovery of fused 5,6-bicyclic heterocycles as γ-secretase modulators
저자
by
Qin, Jun
;
Dhondi, Pawan
;
Huang, Xianhai
;
Mandal, Mihirbaran
;
Zhao, Zhiqiang
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2011 21(2):664-669
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7 . Academic Journal
Iminoheterocycles as γ-secretase modulators
저자
by
Caldwell, John P.
;
Bennett, Chad E.
;
McCracken, Troy M.
;
Mazzola, Robert D.
;
Bara, Thomas
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2010 20(18):5380-5384
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7 . Academic Journal
Structure and activity relationships of tartrate-based TACE inhibitors
저자
by
Li, Dansu
;
Popovici-Muller, Janeta
;
Belanger, David B.
;
Caldwell, John
;
Dai, Chaoyang
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2010 20(16):4812-4815
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