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1 . Academic Journal
Structure-activity relationships of tubulysin analogues
저자
by
Courter, Joel R.
;
Hamilton, Joseph Z.
;
Hendrick, Nathaniel R.
;
Zaval, Margo
;
Waight, Andrew B.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 July 2020 30(14)
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7 . Academic Journal
Improving Antibody‐Tubulysin Conjugates through Linker Chemistry and Site‐Specific Conjugation.
저자
by
Hamilton, Joseph Z.
;
Pires, Thomas A.
;
Mitchell, Jamie A.
;
Cochran, Julia H.
;
Emmerton, Kim K.
, et al.
소스
ChemMedChem; 4/8/2021, Vol. 16 Issue 7, p1077-1081, 5p
Web of Science
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7 . Periodical
Lactone Stabilization is Not a Necessary Feature for Antibody Conjugates of Camptothecins
저자
by
Lau, Uland Y.
;
Benoit, Lauren T.
;
Stevens, Nicole S.
;
Emmerton, Kim K.
;
Zaval, Margo
, et al.
소스
Molecular Pharmaceutics; July 2018, Vol. 15 Issue: 9 p4063-4072, 10p
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7 . Academic Journal
Front Cover: Improving Antibody‐Tubulysin Conjugates through Linker Chemistry and Site‐Specific Conjugation (ChemMedChem 7/2021).
저자
by
Hamilton, Joseph Z.
;
Pires, Thomas A.
;
Mitchell, Jamie A.
;
Cochran, Julia H.
;
Emmerton, Kim K.
, et al.
소스
ChemMedChem; 4/8/2021, Vol. 16 Issue 7, p1047-1047, 1p
Web of Science
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7 . Academic Journal
Discovery of a tripeptide-based camptothecin drug-linker for antibody-drug conjugates with potent antitumor activity and a broad therapeutic window
저자
by
Lyski, Ryan
;
Bou, Lauren
;
Zaval, Margo
;
Emmerton, Kim
;
Okeley, Nicole
, et al.
소스
CANCER RESEARCH
; AUG 2020, 80 16, 2p. Supplement: S
Full Text (AACR)
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7 . Academic Journal
Enfortumab vedotin, an anti-Nectin-4 ADC demonstrates bystander cell killing and immunogenic cell death anti-tumor activity mechanisms of action in urothelial cancers
저자
by
Liu, Bernard A.
;
Olson, Devra
;
Snead, Katie
;
Gosink, John
;
Tenn, Elena-Marie
, et al.
소스
CANCER RESEARCH
; AUG 2020, 80 16, 2p. Supplement: S
Full Text (AACR)
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7 . Academic Journal
Tucatinib, a HER2-selective tyrosine kinase inhibitor, increases the anti-tumor activity of trastuzumab antibody-drug conjugates in preclinical models of HER2+breast cancer
저자
by
Kulukian, Anita
;
Taylor, Janelle
;
Olson, Devra
;
Zaval, Margo
;
Thurman, Robert
, et al.
소스
CANCER RESEARCH
; FEB 2020, 80 4, 2p. Supplement: S
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7 . Academic Journal
Targeted delivery of cytotoxic NAMPT inhibitors using antibody-drug conjugates
저자
by
Neumann, Christopher S.
;
Olivas, Kathleen C.
;
Waight, Andrew B.
;
Meyer, David
;
Loftus, Luke V.
, et al.
소스
CANCER RESEARCH
; JUL 2018, 78 13, 2p. Supplement: S
Full Text (AACR)
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7 . Academic Journal
Additional mechanisms of action of SGN-CD48A in multiple myeloma and improved antitumor activity in combination with daratumumab
저자
by
Olson, Devra J.
;
Liu, Bernard A.
;
Zaval, Margo
;
Cao, Anthony
;
Gurgel, Jesse
, et al.
소스
CANCER RESEARCH
; JUL 2018, 78 13, 2p. Supplement: S
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7 . Academic Journal
Novel auristatins with high activity on efflux-positive models and demonstrable bystander activity
저자
by
Moquist, Philip N.
;
Bovee, Tim D.
;
Waight, Andrew B.
;
Owen, Sarah
;
Mitchell, Jamie A.
, et al.
소스
CANCER RESEARCH
; JUL 2018, 78 13, 1p. Supplement: S
Full Text (AACR)
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