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1 . Academic Journal
AC220 is a uniquely potent and selective inhibitor of FLT3 for the treatment of acute myeloid leukemia (AML)
저자
by
Zarrinkar, Patrick P.
;
Gunawardane, Ruwanthi N.
;
Cramer, Merryl D.
;
Gardner, Michael F.
;
Brigham, Daniel
, et al.
소스
In
Blood
1 October 2009 114(14):2984-2992
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7 . Academic Journal
Discovery and optimization of a highly efficacious class of 5-aryl-2-aminopyridines as FMS-like tyrosine kinase 3 (FLT3) inhibitors
저자
by
Liu, Gang
;
Abraham, Sunny
;
Liu, Xing
;
Xu, Shimin
;
Rooks, Allison M.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 September 2015 25(17):3436-3441
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7 . Academic Journal
Arylcarboxyamino-substituted diaryl ureas as potent and selective FLT3 inhibitors
저자
by
Patel, Hitesh K.
;
Grotzfeld, Robert M.
;
Lai, Andiliy G.
;
Mehta, Shamal A.
;
Milanov, Zdravko V.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2009 19(17):5182-5185
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7 . Academic Journal
Outlier analysis of functional genomic profiles enriches for oncology targets and enables precision medicine.
저자
by
Zhou Zhu
;
Ihle, Nathan T.
;
Rejto, Paul A.
;
Zarrinkar, Patrick P.
.
소스
BMC Genomics
. 6/13/2016, Vol. 17, p1-13. 13p. 2 Charts, 2 Graphs.
Open Access (BioMed Central)
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6 . Academic Journal
The reactivity-driven biochemical mechanism of covalent KRAS
G12C
inhibitors
저자
by
Hansen, Rasmus
;
Peters, Ulf
;
Babbar, Anjali
;
Chen, Yuching
;
Feng, Jun
, et al.
소스
Nature Structural & Molecular Biology
. 25(6):454-462
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7 . Academic Journal
Phase 1 AML Study of AC220, a Potent and Selective Second Generation FLT3 Receptor Tyrosine Kinase Inhibitor
저자
by
Cortes, Jorge E.
;
Ghirdaladze, Darejan
;
Foran, James M.
;
DeVetten, Marcel P.
;
Zodelava, Mamia
, et al.
소스
In
Blood
16 November 2008 112(11):767-767
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7 . Academic Journal
Human Pharmacokinetics of AC220, a Potent and Selective Class III Receptor Tyrosine Kinase Inhibitor.
저자
by
Cortes, Jorge
;
Foran, James M.
;
Devetten, Marcel P.
;
Giles, Francis J.
;
James, Joyce
, et al.
소스
In
Blood
16 November 2007 110(11):1597-1597
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7 . Academic Journal
An Internally Controlled Quantitative Target Occupancy Assay for Covalent Inhibitors
저자
by
Hansen, Rasmus
;
Firdaus, Sarah J.
;
Li, Shuangwei
;
Janes, Matthew R.
;
Zhang, Jingchuan
, et al.
소스
SCIENTIFIC REPORTS
; SEP 25 2018, 8 p14312 7p.
Scopus
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7 . Academic Journal
Validation of ITD mutations in FLT3 as a therapeutic target in human acute myeloid leukaemia
저자
by
Smith, Catherine C.
;
Wang, Qi
;
Chin, Chen-Shan
;
Salerno, Sara
;
Damon, Lauren E.
, et al.
소스
Nature
. May 10, 2012 485(7397):260-263
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7 . Academic Journal
Activation State-Dependent Binding of Small Molecule Kinase Inhibitors: Structural Insights from Biochemistry
저자
by
Wodicka, Lisa M.
;
Ciceri, Pietro
;
Davis, Mindy I.
;
Hunt, Jeremy P.
;
Floyd, Mark
, et al.
소스
Chemistry & Biology
. Nov2010, Vol. 17 Issue 11, p1241-1249. 9p.
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