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1 .
Abstract 1140: A novel MTA non-competitive PRMT5 inhibitor
저자
by
Matt Soars
;
Lisa M. Kopcho
;
Carolyn A. Weigelt
;
Shilpa Demes
;
Gregory D. Vite
, et al.
소스
Cancer Research
. 81:1140-1140
Full Text (AACR)
Web of Science
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7 .
Identification and optimization of a novel series of indoleamine 2,3-dioxygenase inhibitors
저자
by
Steven P. Seitz
;
John T. Hunt
;
Kelly L. Covello
;
Lisa Elkin
;
Gregory D. Vite
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 27:582-585
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7 .
Identification of imidazo[1,2-b]pyridazine TYK2 pseudokinase ligands as potent and selective allosteric inhibitors of TYK2 signalling
저자
by
Dianlin Xie
;
Jing Chen
;
Celia D’Arienzo
;
Jodi K. Muckelbauer
;
Nelly Aranibar
, et al.
소스
MedChemComm
. 8:700-712
Open Access (OpenAIRE)
Scopus
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7 .
Building homogeneous time-resolved fluorescence resonance energy transfer assays for characterization of bivalent inhibitors of an inhibitor of apoptosis protein target
저자
by
Litao Zhang
;
William J. Metzler
;
Shana L. Posy
;
Robert M. Borzilleri
;
Yuval Blat
, et al.
소스
Analytical Biochemistry
. 497:8-17
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7 .
Tyrosine Kinase 2-mediated Signal Transduction in T Lymphocytes Is Blocked by Pharmacological Stabilization of Its Pseudokinase Domain
저자
by
Stephen R. Johnson
;
Dianlin Xie
;
Lihong Cheng
;
Yang Hong
;
John S. Tokarski
, et al.
소스
Journal of Biological Chemistry
. 290:11061-11074
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7 .
Structure activity relationship studies on chemically non-reactive glycine sulfonamide inhibitors of diacylglycerol lipase
저자
by
Martin A. Lewis
;
Louis S. Chupak
;
Robert G. Gentles
;
Shuanghua Hu
;
Min Ding
, et al.
소스
Bioorganicmedicinal chemistry
. 24(7)
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7 .
Postsynaptic diacylglycerol lipase α mediates retrograde endocannabinoid suppression of inhibition in mouse prefrontal cortex
저자
by
Brian Zambrowicz
;
Ryan Westphal
;
David A. Lewis
;
Donna L. Pedicord
;
Michael J. Flynn
, et al.
소스
The Journal of Physiology
. 589:4857-4884
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7 .
An electrophoretic mobility shift assay for the identification and kinetic analysis of acetyl transferase inhibitors
저자
by
Donna L. Pedicord
;
Sujatha Nagulapalli
;
Caroline Fanslau
;
Lata Jayaraman
;
Jonathan Lippy
, et al.
소스
Analytical Biochemistry
. 402:65-68
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7 .
Non-Competitive Inhibition by Active Site Binders
저자
by
Yuval Blat
.
소스
Chemical Biology & Drug Design
. 75:535-540
Open Access (OpenAIRE)
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3 .
The Amyloid-β Rise and γ-Secretase Inhibitor Potency Depend on the Level of Substrate Expression
저자
by
Bergstrom Carl P
;
Jeremy H. Toyn
;
Robert H. Grafstrom
;
Yang Michael G
;
Mcelhone Katharine E
, et al.
소스
Journal of Biological Chemistry
. 283:22992-23003
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