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1 . Periodical
Optimization of Potent, Selective, and Orally Bioavailable Pyrrolodinopyrimidine-Containing Inhibitors of Heat Shock Protein 90. Identification of Development Candidate 2-Amino-4-{4-chloro-2-[2-(4-fluoro-1H-pyrazol-1-yl)ethoxy]-6-methylphenyl}-N-(2,2-difluoropropyl)-5,7-dihydro-6H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
저자
by
Zehnder, Luke
;
Bennett, Michael
;
Meng, Jerry
;
Huang, Buwen
;
Ninkovic, Sacha
, et al.
소스
Journal of Medicinal Chemistry; 20240101, Issue: Preprints
Full Text (ACS)
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7 . Academic Journal
Conformationally-restricted cyclic sulfones as potent and selective mTOR kinase inhibitors
저자
by
Liu, Kevin K.-C.
;
Bailey, Simon
;
Dinh, Dac M.
;
Lam, Hieu
;
Li, Chunze
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 August 2012 22(15):5114-5117
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7 . Academic Journal
Dihydroxylphenyl amides as inhibitors of the Hsp90 molecular chaperone
저자
by
Kung, Pei-Pei
;
Funk, Lee
;
Meng, Jerry
;
Collins, Michael
;
Zhou, Joe Zhongxiang
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 December 2008 18(23):6273-6278
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7 . Academic Journal
Suppression of Heat Shock Protein 27 Using OGX-427 Induces Endoplasmic Reticulum Stress and Potentiates Heat Shock Protein 90 Inhibitors to Delay Castrate-resistant Prostate Cancer.
저자
by
Lamoureux, François
;
Thomas, Christian
;
Yin, Min-Jean
;
Fazli, Ladan
;
Zoubeidi, Amina
, et al.
소스
European Urology
. Jul2014, Vol. 66 Issue 1, p145-155. 11p.
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7 . Academic Journal
miR-122 Regulates Tumorigenesis in Hepatocellular Carcinoma by Targeting AKT3.
저자
by
Nassirpour, Rounak
;
Mehta, Pramod P.
;
Yin, Min-Jean
.
소스
PLoS ONE
. Nov2013, Vol. 8 Issue 11, p1-10. 10p.
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5 . Academic Journal
miR-221 Promotes Tumorigenesis in Human Triple Negative Breast Cancer Cells.
저자
by
Nassirpour, Rounak
;
Mehta, Pramod P.
;
Baxi, Sangita M.
;
Yin, Min-Jean
.
소스
PLoS ONE
. Apr2013, Vol. 8 Issue 4, p1-9. 9p.
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6 . Academic Journal
Clusterin Inhibition Using OGX-011 Synergistically Enhances Hsp90 Inhibitor Activity by Suppressing the Heat Shock Response in Castrate-Resistant Prostate Cancer.
저자
by
Lamoureux, Francois
;
Thomas, Christian
;
Yin, Min-Jean
;
Kuruma, Hidetoshi
;
Beraldi, Eliana
, et al.
소스
Cancer Research
. Sep2011, Vol. 71 Issue 17, p5838-5849. 12p.
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7 . Academic Journal
Optimization of Potent, Selective, and Orally Bioavailable Pyrrolodinopyrimidine-Containing Inhibitors of Heat Shock Protein 90. Identification of Development Candidate 2-Amino-4-{4-chloro-2-[2-(4-fluoro-1H-pyrazol-1-yl)ethoxy]-6-methylphenyl}-N-(2,2-difluoropropyl)-5,7-dihydro-6H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
저자
by
Zehnder, Luke
;
Bennett, Michael
;
Meng, Jerry
;
Huang, Buwen
;
Ninkovic, Sacha
, et al.
소스
Journal of Medicinal Chemistry
. 5/12/2011, Vol. 54 Issue 9, p3368-3385. 18p.
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7 . Academic Journal
RETRACTED: A novel class of specific Hsp90 small molecule inhibitors demonstrate in vitro and in vivo anti-tumor activity in human melanoma cells.
저자
by
Mehta PP
;
Kung PP
;
Yamazaki S
;
Walls M
;
Shen A
, et al.
소스
Cancer Letters
. Jan2011, Vol. 300 Issue 1, p30-39. 10p.
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7 . Academic Journal
A novel class of specific Hsp90 small molecule inhibitors demonstrate in vitro and in vivo anti-tumor activity in human melanoma cells
저자
by
Mehta, Pramod P.
;
Kung, Pei-Pei
;
Yamazaki, Shinji
;
Walls, Marlena
;
Shen, Andrea
, et al.
소스
Cancer Letters
. Jan2011, Vol. 300 Issue 1, p30-39. 10p.
Full Text (Clinical Key)
Full Text (ScienceDirect)
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