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1 . Academic Journal
Design and optimisation of dendrimer-conjugated Bcl-2/xL inhibitor, AZD0466, with improved therapeutic index for cancer therapy
저자
by
Claire M. Patterson
;
Srividya B. Balachander
;
Iain Grant
;
Petar Pop-Damkov
;
Brian Kelly
, et al.
소스
Communications Biology, Vol 4, Iss 1, Pp 1-14 (2021)
Open Access (DOAJ)
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7 . Academic Journal
The acute glucose lowering effect of specific GPR120 activation in mice is mainly driven by glucagon-like peptide 1.
저자
by
Linda Sundström
;
Susanna Myhre
;
Monika Sundqvist
;
Andrea Ahnmark
;
William McCoull
, et al.
소스
PLoS ONE, Vol 12, Iss 12, p e0189060 (2017)
Open Access (DOAJ)
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7 .
Figure S6 from AZD4320, A Dual Inhibitor of Bcl-2 and Bcl-xL, Induces Tumor Regression in Hematologic Cancer Models without Dose-limiting Thrombocytopenia
저자
by
Francis D. Gibbons
;
Stephen E. Fawell
;
Barry R. Davies
;
J. Paul Secrist
;
Michael Zinda
, et al.
소스
Open Access (OpenAIRE)
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7 .
Supplementary Data_Clean from AZD4320, A Dual Inhibitor of Bcl-2 and Bcl-xL, Induces Tumor Regression in Hematologic Cancer Models without Dose-limiting Thrombocytopenia
저자
by
Francis D. Gibbons
;
Stephen E. Fawell
;
Barry R. Davies
;
J. Paul Secrist
;
Michael Zinda
, et al.
소스
Open Access (OpenAIRE)
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7 .
Data from AZD4320, A Dual Inhibitor of Bcl-2 and Bcl-xL, Induces Tumor Regression in Hematologic Cancer Models without Dose-limiting Thrombocytopenia
저자
by
Francis D. Gibbons
;
Stephen E. Fawell
;
Barry R. Davies
;
J. Paul Secrist
;
Michael Zinda
, et al.
소스
Open Access (OpenAIRE)
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7 .
Pharmacological inhibition of MERTK induces in vivo retinal degeneration: a multimodal imaging ocular safety assessment
저자
by
Gregory Hamm
;
Gareth Maglennon
;
Beth Williamson
;
Ruth Macdonald
;
Ann Doherty
, et al.
소스
Archives of Toxicology
. 96:613-624
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7 .
Optimization of an Imidazo[1,2-a]pyridine Series to Afford Highly Selective Type I1/2 Dual Mer/Axl Kinase Inhibitors with In Vivo Efficacy
저자
by
Edward J. Hennessy
;
Marianne Schimpl
;
Emma Rivers
;
Paul D. Smith
;
Elizabeth Hardaker
, et al.
소스
Journal of Medicinal Chemistry
. 64:13524-13539
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7 .
Identification and Strategies to Mitigate High Total Clearance of Benzylamine-Substituted Biphenyl Ring Systems
저자
by
Beth Williamson
;
Lindsay McMurray
;
Scott Boyd
;
Olga Collingwood
;
Neville McLean
, et al.
소스
Molecular pharmaceutics
. 19(7)
Scopus
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7 .
Diversity-orientated synthesis of macrocyclic heterocycles using a double SNAr approach
저자
by
Morgan Thomas
;
Piotr Raubo
;
Rodrigo J. Carbajo
;
Joanna Raubo
;
William McCoull
.
소스
Organic & Biomolecular Chemistry
. 19:6274-6290
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7 .
AZD4320, A Dual Inhibitor of Bcl-2 and Bcl-xL, Induces Tumor Regression in Hematologic Cancer Models without Dose-limiting Thrombocytopenia
저자
by
Shenghua Wen
;
Srividya B. Balachander
;
Francis D. Gibbons
;
Michael Zinda
;
William McCoull
, et al.
소스
Clinical Cancer Research
. 26:6535-6549
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