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1 . Academic Journal
Multifunctional agents against Alzheimer’s disease based on oxidative stress: Polysubstituted pyrazine derivatives synthesized by multicomponent reactions
저자
by
Wei, Wenxiu
;
Jing, Lanlan
;
Tian, Ye
;
Więckowska, Anna
;
Kang, Dongwei
, et al.
소스
In
Bioorganic & Medicinal Chemistry
15 December 2023 96
Full Text (ScienceDirect)
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7 . Academic Journal
Novel drug-like fluorenyl derivatives as selective butyrylcholinesterase and β-amyloid inhibitors for the treatment of Alzheimer’s disease
저자
by
Pasieka, Anna
;
Panek, Dawid
;
Zaręba, Paula
;
Sługocka, Emilia
;
Gucwa, Natalia
, et al.
소스
In
Bioorganic & Medicinal Chemistry
6 June 2023 88-89
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7 . Academic Journal
Discovery of new, highly potent and selective inhibitors of BuChE - design, synthesis, in vitro and in vivo evaluation and crystallography studies
저자
by
Panek, Dawid
;
Pasieka, Anna
;
Latacz, Gniewomir
;
Zaręba, Paula
;
Szczęch, Michał
, et al.
소스
In
European Journal of Medicinal Chemistry
5 March 2023 249
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7 . Academic Journal
Bacterial type I signal peptidase inhibitors - Optimized hits from nature
저자
by
Szałaj, Natalia
;
Benediktsdottir, Andrea
;
Rusin, Dominika
;
Karlén, Anders
;
Mowbray, Sherry L.
, et al.
소스
In
European Journal of Medicinal Chemistry
5 August 2022 238
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7 . Academic Journal
Development and crystallography-aided SAR studies of multifunctional BuChE inhibitors and 5-HT6R antagonists with β-amyloid anti-aggregation properties
저자
by
Wichur, Tomasz
;
Godyń, Justyna
;
Góral, Izabella
;
Latacz, Gniewomir
;
Bucki, Adam
, et al.
소스
In
European Journal of Medicinal Chemistry
5 December 2021 225
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7 . Academic Journal
Discovery of 1-(phenylsulfonyl)-1H-indole-based multifunctional ligands targeting cholinesterases and 5-HT6 receptor with anti-aggregation properties against amyloid-beta and tau
저자
by
Wichur, Tomasz
;
Pasieka, Anna
;
Godyń, Justyna
;
Panek, Dawid
;
Góral, Izabella
, et al.
소스
In
European Journal of Medicinal Chemistry
5 December 2021 225
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7 . Academic Journal
Discovery of multifunctional anti-Alzheimer’s agents with a unique mechanism of action including inhibition of the enzyme butyrylcholinesterase and γ-aminobutyric acid transporters
저자
by
Pasieka, Anna
;
Panek, Dawid
;
Jończyk, Jakub
;
Godyń, Justyna
;
Szałaj, Natalia
, et al.
소스
In
European Journal of Medicinal Chemistry
5 June 2021 218
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7 . Academic Journal
1-Benzylpyrrolidine-3-amine-based BuChE inhibitors with anti-aggregating, antioxidant and metal-chelating properties as multifunctional agents against Alzheimer’s disease
저자
by
Wichur, Tomasz
;
Więckowska, Anna
;
Więckowski, Krzysztof
;
Godyń, Justyna
;
Jończyk, Jakub
, et al.
소스
In
European Journal of Medicinal Chemistry
1 February 2020 187
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7 . Academic Journal
Design, synthesis and biological evaluation of new phthalimide and saccharin derivatives with alicyclic amines targeting cholinesterases, beta-secretase and amyloid beta aggregation
저자
by
Panek, Dawid
;
Więckowska, Anna
;
Wichur, Tomasz
;
Bajda, Marek
;
Godyń, Justyna
, et al.
소스
In
European Journal of Medicinal Chemistry
5 January 2017 125:676-695
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7 . Academic Journal
Connecting GSK-3β Inhibitory Activity with IKK-β or ROCK-1 Inhibition to Target Tau Aggregation and Neuroinflammation in Alzheimer's Disease—Discovery, In Vitro and In Cellulo Activity of Thiazole-Based Inhibitors.
저자
by
Góral, Izabella
;
Wichur, Tomasz
;
Sługocka, Emilia
;
Godyń, Justyna
;
Szałaj, Natalia
, et al.
소스
Molecules
. Jun2024, Vol. 29 Issue 11, p2616. 32p.
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