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1 . Academic Journal
The Plasmodium falciparum ABC transporter ABCI3 confers parasite strain-dependent pleiotropic antimalarial drug resistance
저자
by
Murithi, James M.
;
Deni, Ioanna
;
Pasaje, Charisse Flerida A.
;
Okombo, John
;
Bridgford, Jessica L.
, et al.
소스
In
Cell Chemical Biology
19 May 2022 29(5):824-839
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7 . Academic Journal
Inhibition of Resistance-Refractory P. falciparum Kinase PKG Delivers Prophylactic, Blood Stage, and Transmission-Blocking Antiplasmodial Activity
저자
by
Vanaerschot, Manu
;
Murithi, James M.
;
Pasaje, Charisse Flerida A.
;
Ghidelli-Disse, Sonja
;
Dwomoh, Louis
, et al.
소스
In
Cell Chemical Biology
16 July 2020 27(7):806-816
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7 . Academic Journal
hERG, Plasmodium Life Cycle, and Cross Resistance Profiling of New Azabenzimidazole Analogues of Astemizole.
저자
by
Mambwe, Dickson
;
Coertzen, Dina
;
Leshabane, Meta
;
Mulubwa, Mwila
;
Njoroge, Mathew
, et al.
소스
ACS Medicinal Chemistry Letters; 4/11/2024, Vol. 15 Issue 4, p463-469, 7p
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7 . Academic Journal
Bayesian models trained with HTS data for predicting β-haematin inhibition and in vitro antimalarial activity
저자
by
Wicht, Kathryn J.
;
Combrinck, Jill M.
;
Smith, Peter J.
;
Egan, Timothy J.
.
소스
In
Bioorganic & Medicinal Chemistry
15 August 2015 23(16):5210-5217
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6 . Academic Journal
N10,N11-di-alkylamine indolo[3,2-b]quinolines as hemozoin inhibitors: Design, synthesis and antiplasmodial activity
저자
by
Figueiras, Marta
;
Coelho, Lis
;
Wicht, Kathryn J.
;
Santos, Sofia A.
;
Lavrado, João
, et al.
소스
In
Bioorganic & Medicinal Chemistry
1 April 2015 23(7):1530-1539
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7 . Academic Journal
Drug discovery in Africa tackles zoonotic and related infections.
저자
by
Hikaambo, Christabel N.
;
Shakela, Natalia
;
Woodland, John G.
;
Wicht, Kathryn J.
;
Chibale, Kelly
.
소스
Science Translational Medicine; 10/18/2023, Vol. 15 Issue 718, p1-5, 5p
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7 . Academic Journal
Identification of β-hematin inhibitors in a high-throughput screening effort reveals scaffolds with in vitro antimalarial activity
저자
by
Sandlin, Rebecca D.
;
Fong, Kim Y.
;
Wicht, Kathryn J.
;
Carrell, Holly M.
;
Egan, Timothy J.
, et al.
소스
In
International Journal for Parasitology: Drugs and Drug Resistance
December 2014 4(3):316-325
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7 . Academic Journal
Synthesis, β-haematin inhibition, and in vitro antimalarial testing of isocryptolepine analogues: SAR study of indolo[3,2-c]quinolines with various substituents at C2, C6, and N11
저자
by
Wang, Ning
;
Wicht, Kathryn J.
;
Imai, Kento
;
Wang, Ming-qi
;
Anh Ngoc, Tran
, et al.
소스
In
Bioorganic & Medicinal Chemistry
1 May 2014 22(9):2629-2642
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7 . Academic Journal
In vitro antimalarial activity, β-haematin inhibition and structure–activity relationships in a series of quinoline triazoles
저자
by
Joshi, Mukesh C.
;
Wicht, Kathryn J.
;
Taylor, Dale
;
Hunter, Roger
;
Smith, Peter J.
, et al.
소스
In
European Journal of Medicinal Chemistry
November 2013 69:338-347
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7 . Academic Journal
Synthesis and antimalarial testing of neocryptolepine analogues: Addition of ester function in SAR study of 2,11-disubstituted indolo[2,3-b]quinolines
저자
by
Lu, Wen-Jie
;
Wicht, Kathryn J.
;
Wang, Li
;
Imai, Kento
;
Mei, Zhen-Wu
, et al.
소스
In
European Journal of Medicinal Chemistry
June 2013 64:498-511
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