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1 . Academic Journal
Discovery of first-in-class multi-target adenosine A2A receptor antagonists-carbonic anhydrase IX and XII inhibitors. 8-Amino-6-aryl-2-phenyl-1,2,4-triazolo [4,3-a]pyrazin-3-one derivatives as new potential antitumor agents
저자
by
Ceni, Costanza
;
Catarzi, Daniela
;
Varano, Flavia
;
Ben, Diego Dal
;
Marucci, Gabriella
, et al.
소스
In
European Journal of Medicinal Chemistry
1 September 2020 201
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7 . Academic Journal
Anticancer activity study of A3 adenosine receptor agonists
저자
by
Marucci, Gabriella
;
Santinelli, Claudia
;
Buccioni, Michela
;
Navia, Aleix Martí
;
Lambertucci, Catia
, et al.
소스
In
Life Sciences
15 July 2018 205:155-163
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7 . Academic Journal
New potent and selective A1 adenosine receptor antagonists as potential tools for the treatment of gastrointestinal diseases
저자
by
Lambertucci, Catia
;
Marucci, Gabriella
;
Dal Ben, Diego
;
Buccioni, Michela
;
Spinaci, Andrea
, et al.
소스
In
European Journal of Medicinal Chemistry
10 May 2018 151:199-213
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7 . Academic Journal
Structural Investigations on 2-Amidobenzimidazole Derivatives as New Inhibitors of Protein Kinase CK1 Delta.
저자
by
Calenda, Sara
;
Catarzi, Daniela
;
Varano, Flavia
;
Vigiani, Erica
;
Volpini, Rosaria
, et al.
소스
Pharmaceuticals (14248247)
. Apr2024, Vol. 17 Issue 4, p468. 31p.
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7 . Academic Journal
Adenine derivatives as inhibitors of the casein kinase CK1delta enzyme.
저자
by
Spinaci, Andrea
;
Lambertucci, Catia
;
Chang, Cui
;
Buccioni, Michela
;
Marucci, Gabriella
, et al.
소스
Medicinal Chemistry Research; Apr2024, Vol. 33 Issue 4, p611-619, 9p
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7 . Academic Journal
Exploring the 2- and 5-positions of the pyrazolo[4,3-d]pyrimidin-7-amino scaffold to target human A1 and A2A adenosine receptors
저자
by
Squarcialupi, Lucia
;
Falsini, Matteo
;
Catarzi, Daniela
;
Varano, Flavia
;
Betti, Marco
, et al.
소스
In
Bioorganic & Medicinal Chemistry
15 June 2016 24(12):2794-2808
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7 . Academic Journal
Exploring the 7-oxo-thiazolo[5,4-d]pyrimidine core for the design of new human adenosine A3 receptor antagonists. Synthesis, molecular modeling studies and pharmacological evaluation
저자
by
Varano, Flavia
;
Catarzi, Daniela
;
Squarcialupi, Lucia
;
Betti, Marco
;
Vincenzi, Fabrizio
, et al.
소스
In
European Journal of Medicinal Chemistry
26 May 2015 96:105-121
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7 . Academic Journal
Purinergic P2X receptors: Structural models and analysis of ligand-target interaction
저자
by
Dal Ben, Diego
;
Buccioni, Michela
;
Lambertucci, Catia
;
Marucci, Gabriella
;
Thomas, Ajiroghene
, et al.
소스
In
European Journal of Medicinal Chemistry
7 January 2015 89:561-580
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7 . Academic Journal
1,2,4-Triazolo[1,5-a]quinoxaline derivatives and their simplified analogues as adenosine A3 receptor antagonists. Synthesis, structure–affinity relationships and molecular modeling studies
저자
by
Catarzi, Daniela
;
Varano, Flavia
;
Poli, Daniela
;
Squarcialupi, Lucia
;
Betti, Marco
, et al.
소스
In
Bioorganic & Medicinal Chemistry
1 January 2015 23(1):9-21
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7 . Academic Journal
8-(2-Furyl)adenine derivatives as A2A adenosine receptor ligands
저자
by
Dal Ben, Diego
;
Buccioni, Michela
;
Lambertucci, Catia
;
Thomas, Ajiroghene
;
Klotz, Karl-Norbert
, et al.
소스
In
European Journal of Medicinal Chemistry
December 2013 70:525-535
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