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1 . Academic Journal
Ketorolac modulates Rac-1/HIF-1α/DDX3/β-catenin signalling via a tumor suppressor prostate apoptosis response-4 (Par-4) in renal cell carcinoma
저자
by
Vinay Sonawane
;
Jeevan Ghosalkar
;
Swati Achrekar
;
Kalpana Joshi
.
소스
Scientific Reports, Vol 13, Iss 1, Pp 1-15 (2023)
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6 . Academic Journal
Prostate Apoptosis Response-4 (Par-4): A Novel Target in Pyronaridine-Induced Apoptosis in Glioblastoma (GBM) Cells
저자
by
Jeevan Ghosalkar
;
Vinay Sonawane
;
Tejal Pisal
;
Swati Achrekar
;
Radha Pujari
, et al.
소스
Cancers, Vol 14, Iss 13, p 3198 (2022)
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7 .
Furanoflavones pongapin and lanceolatin B blocks the cell cycle and induce senescence in CYP1A1-overexpressing breast cancer cells
저자
by
Sandip B. Bharate
;
Linda Gatchie
;
Bhabatosh Chaudhuri
;
Ibidapo S. Williams
;
Rajni Sharma
, et al.
소스
Bioorganic & Medicinal Chemistry
. 26:6076-6086
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7 .
Prostate Apoptosis Response-4: a Therapeutic Target for Malignant Gliomas
저자
by
Jeevan Ghosalkar
;
Vinay Sonawane
;
Mohsina Khan
;
Kalpana Joshi
;
Padma Shastry
.
소스
Tumor Suppressor Par-4 ISBN: 9783030805579
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7 .
Khellinoflavanone, a Semisynthetic Derivative of Khellin, Overcomes Benzo[a]pyrene Toxicity in Human Normal and Cancer Cells That Express CYP1A1
저자
by
Linda Gatchie
;
Ibidapo S. Williams
;
Bhabatosh Chaudhuri
;
Rajni Sharma
;
Sandip B. Bharate
, et al.
소스
ACS Omega, Vol 3, Iss 8, Pp 8553-8566 (2018)
ACS Omega
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7 .
Identification of Potent and Selective CYP1A1 Inhibitors via Combined Ligand and Structure-Based Virtual Screening and Their in Vitro Validation in Sacchrosomes and Live Human Cells
저자
by
Vinay Sonawane
;
Prashant Joshi
;
Ram A. Vishwakarma
;
Glen J. P. McCann
;
Sandip B. Bharate
, et al.
소스
Journal of Chemical Information and Modeling
. 57:1309-1320
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7 .
Cink4T, a quinazolinone-based dual inhibitor of Cdk4 and tubulin polymerization, identified via ligand-based virtual screening, for efficient anticancer therapy
저자
by
Bhabatosh Chaudhuri
;
Venkatesan Jayaprakash
;
Barij Nayan Sinha
;
Surender Singh Jadav
;
Vinay Sonawane
, et al.
소스
European journal of medicinal chemistry
. 165
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7 .
CYP enzymes, expressed within live human suspension cells, are superior to widely-used microsomal enzymes in identifying potent CYP1A1/CYP1B1 inhibitors: Identification of quinazolinones as CYP1A1/CYP1B1 inhibitors that efficiently reverse B[a]P toxicity and cisplatin resistance
저자
by
Barij Nayan Sinha
;
Mohd Usman Mohd Siddique
;
Bhabatosh Chaudhuri
;
Ibidapo S. Williams
;
Sandip B. Bharate
, et al.
소스
European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences
. 131
Open Access (OpenAIRE)
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7 .
Identification of karanjin isolated from the Indian beech tree as a potent CYP1 enzyme inhibitor with cellular efficacy via screening of a natural product repository
저자
by
Sandip B. Bharate
;
Bhabatosh Chaudhuri
;
Naresh Kumar Satti
;
Rajni Sharma
;
Glen J. P. McCann
, et al.
소스
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7 .
(E)-3-(3,4,5-Trimethoxyphenyl)-1-(pyridin-4-yl)prop-2-en-1-one, a heterocyclic chalconeis a potent and selectiveCYP1A1 inhibitor and cancerchemopreventative agent
저자
by
Kenneth J. M. Beresford
;
Supriya Kaduskar
;
Linda Gatchie
;
Prashant Joshi
;
Vinay Sonawane
, et al.
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