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1 . Academic Journal
Preclinical efficacy of the potent, selective menin-KMT2A inhibitor JNJ-75276617 (bleximenib) in KMT2A- and NPM1-altered leukemias
저자
by
Kwon, Min Chul
;
Thuring, Jan Willem
;
Querolle, Olivier
;
Dai, Xuedong
;
Verhulst, Tinne
, et al.
소스
In
Blood
12 September 2024 144(11):1206-1220
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7 . Academic Journal
Pharmacological Characterization of JNJ-75276617, a Menin-KMT2A Inhibitor, As Targeted Treatment for KMT2A-Altered and NPM1-Mutant Acute Leukemia
저자
by
Kwon, Min Chul
;
Querolle, Olivier
;
Dai, Xuedong
;
Thuring, Jan Willem
;
Verhulst, Tinne
, et al.
소스
In
Blood
15 November 2022 140 Supplement 1:5928-5929
Full Text (ScienceDirect)
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7 . Periodical
Discovery of a Novel, First-in-Class Bfl-1 BH3 Mimetic with Pro-Apoptotic Activity
저자
by
Derks, Maarten
;
Bryan, Marian C.
;
Rockx, Cindy
;
Schults, Tamara
;
Verhulst, Tinne
, et al.
소스
Blood; November 2023, Vol. 142 Issue: 1, Number 1 Supplement 1 p2824-2824, 1p
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7 . Periodical
Preclinical Efficacy of the Menin-KMT2A Inhibitor JNJ-75276617 in Combination with Venetoclax and Azacitidine in AML
저자
by
Kwon, Min Chul
;
Verhulst, Tinne
;
Goffin, Dries
;
Marien, Ann
;
Verbist, Bie
, et al.
소스
Blood; November 2023, Vol. 142 Issue: 1, Number 1 Supplement 1 p4167-4167, 1p
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7 . Academic Journal
Interleukin-6 is a potential therapeutic target in interleukin-6 dependent, estrogen receptor-α-positive breast cancer.
저자
by
Casneuf, Tineke
;
Axel, Amy E.
;
King, Peter
;
Alvarez, John D.
;
Werbeck, Jillian L.
, et al.
소스
Breast Cancer: Targets & Therapy; Feb2016, Vol. 8, p12-27, 15p
Open Access (T&F)
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7 . Academic Journal
Discovery and Pharmacological Characterization of JNJ-42756493 (Erdafitinib), a Functionally Selective Small-Molecule FGFR Family Inhibitor
저자
by
Perera, Timothy P. S.
;
Jovcheva, Eleonora
;
Mevellec, Laurence
;
Vialard, Jorge
;
De lange, Desiree
, et al.
소스
MOLECULAR CANCER THERAPEUTICS
; JUN 2017, 16 6, p1010-p1020, 11p.
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7 . Academic Journal
Rational combinations with the HDAC inhibitor JNJ-26481585: Prostate cancer and taxane therapy
저자
by
Hickson, Ian
;
King, Peter
;
Marien, Ann
;
Vreys, Veronique
;
Janssen, Marc
, et al.
소스
CANCER RESEARCH
; APR 2010, 70 4p. Supplement: 8
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7 . Academic Journal
Preclinical assessment of the HDAC inhibitor JNJ-26481585: potent in vivo activity across a broad spectrum of human tumor xenografts
저자
by
Hickson, Ian
;
King, Peter
;
Marien, Ann
;
Janssen, Lut
;
Floren, Wim
, et al.
소스
CANCER RESEARCH
; APR 2010, 70 4p. Supplement: 8
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7 . Academic Journal
OMO-1, a potent, highly selective, orally bioavailable, MET kinase inhibitor with a favorable preclinical toxicity profile, shows both monotherapy activity, against MET pathway-driven tumors, and EGFR TKI combination activity in acquired resistance models
저자
by
Libouban, Marion
;
Jovcehva, Eleonora
;
De lange, Desiree
;
Janssens, Boudewijn
;
Verhulst, Tinne
, et al.
소스
CANCER RESEARCH
; JUL 2018, 78 13, 2p. Supplement: S
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7 . Academic Journal
A novel PRMT5 inhibitor with potent in vitro and in vivo activity in preclinical lung cancer models
저자
by
Brehmer, Dirk
;
Wu, Tongfei
;
Mannens, Geert
;
Beke, Lijs
;
Vinken, Petra
, et al.
소스
CANCER RESEARCH
; JUL 2017, 77 2p. Supplement: 13
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