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1 .
Proteopedia entry: Structure of complex membrane proteins solved using cryo-electron microscopy
저자
by
Abby Hillan
;
Emily Neal
;
Shelby Skaggs
;
Carson Middlebrook
;
Daniel Mulawa
, et al.
소스
Biochemistry and molecular biology education : a bimonthly publication of the International Union of Biochemistry and Molecular BiologyREFERENCE
. 49(5)
EBSCOHost PDF
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7 .
Circularly polarized luminescence of
S
m (III) and
E
u (III) complexes with chiral ligand (
R
/
S
)‐
BINAPO
저자
by
Spencer Dodder
;
Valentine J. Klimkowski
;
Daniel Cotter
;
Todd A. Hopkins
.
소스
Chirality
. 31:301-311
Web of Science
Scopus
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6 .
Dual Exosite-binding Inhibitors of Insulin-degrading Enzyme Challenge Its Role as the Primary Mediator of Insulin Clearance in Vivo
저자
by
Timothy B. Durham
;
Jeffrey T. Dixon
;
James Lee Toth
;
Angela M. Siesky
;
Michael E. Christe
, et al.
소스
Journal of Biological Chemistry
. 290:20044-20059
Full Text (ScienceDirect O/A)
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7 .
Identification of Potent and Selective Hydantoin Inhibitors of Aggrecanase-1 and Aggrecanase-2 That Are Efficacious in Both Chemical and Surgical Models of Osteoarthritis
저자
by
C. Lin
;
Chin Liu
;
Valentine J. Klimkowski
;
Craig A. Swearingen
;
Lisa A. Adams
, et al.
소스
Journal of Medicinal Chemistry
. 57:10476-10485
Web of Science
Scopus
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7 .
Metabolic-intermediate complex formation with cytochrome P450: Theoretical studies in elucidating the reaction pathway for the generation of reactive nitroso intermediate
저자
by
Michael A. Mohutsky
;
Valentine J. Klimkowski
;
Bhargav Patel
;
Prasad V. Bharatam
;
Nikhil Taxak
, et al.
소스
Journal of Computational Chemistry
. 33:1740-1747
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7 .
Investigation of the terminal P4 domain in a series of d-phenylglycinamide-based factor Xa inhibitors
저자
by
Gerald F. Smith
;
Wayne W. Weber
;
John Walter Nr Macclesfield Liebeschuetz
;
Philip Sipes
;
Jeffry Bernard Franciskovich
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 17:6910-6913
Web of Science
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7 .
d-Phenylglycinol-derived non-covalent factor Xa inhibitors: Effect of non-peptidic S4 linkage elements on affinity and anticoagulant activity
저자
by
Scott Martin Sheehan
;
Nikolay Y. Chirgadze
;
Gerald F. Smith
;
Jolie Anne Bastian
;
Michael Robert Wiley
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 17:5801-5805
Web of Science
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7 .
Preparation and biological evaluation of conformationally constrained BACE1 inhibitors
저자
by
Stephanie L. Stout
;
Patrick C. May
;
Brian Morgan Watson
;
Pablo Garcia Losada
;
Valentine J. Klimkowski
, et al.
소스
Bioorganicmedicinal chemistry
. 23(13)
Full Text (ScienceDirect)
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Scopus
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7 .
N2-Aroylanthranilamide Inhibitors of Human Factor Xa
저자
by
Linebarger Jh
;
Michael Robert Wiley
;
Leonard C. Weir
;
Trelia J. Craft
;
Goodson T
, et al.
소스
Journal of Medicinal Chemistry
. 43:873-882
Web of Science
Scopus
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7 .
Dibasic benzo[b]thiophene derivatives as a novel class of active site directed thrombin inhibitors: 2: sidechain optimization and demonstration of in vivo efficacy
저자
by
Sau-Chi B. Yan
;
Michael L. Denney
;
Valentine J. Klimkowski
;
Amy J. Smith
;
Lea M. Johnson
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 9:775-780
Web of Science
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