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1 . Academic Journal
Discovery of KB-0742, a Potent, Selective, Orally Bioavailable Small Molecule Inhibitor of CDK9 for MYC-Dependent Cancers.
저자
by
Freeman, David B.
;
Hopkins, Tamara D.
;
Mikochik, Peter J.
;
Vacca, Joseph P.
;
Gao, Hua
, et al.
소스
Journal of Medicinal Chemistry; 12/14/2023, Vol. 66 Issue 23, p15629-15647, 19p
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7 . Academic Journal
Discovery of potent, selective 4-fluoroproline-based thrombin inhibitors with improved metabolic stability
저자
by
Staas, Donnette D.
;
Savage, Kelly L.
;
Sherman, Vanessa L.
;
Shimp, Heidi L.
;
Lyle, Terry A.
, et al.
소스
In
Bioorganic & Medicinal Chemistry
2006 14(20):6900-6916
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7 . Academic Journal
Biochemical and cell-based assays for characterization of BACE-1 inhibitors
저자
by
Pietrak, Beth L.
;
Crouthamel, Ming-Chih
;
Tugusheva, Katherine
;
Lineberger, Janet E.
;
Xu, Min
, et al.
소스
In
Analytical Biochemistry
2005 342(1):144-151
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7 . Academic Journal
Development of macrocyclic inhibitors of HCV NS3/4A protease with cyclic constrained P2–P4 linkers
저자
by
Rudd, Michael T.
;
McIntyre, Charles J.
;
Romano, Joseph J.
;
Butcher, John W.
;
Holloway, M. Katharine
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 December 2012 22(23):7207-7213
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7 . Academic Journal
Development of potent macrocyclic inhibitors of genotype 3a HCV NS3/4A protease
저자
by
Rudd, Michael T.
;
McCauley, John A.
;
Romano, Joseph J.
;
Butcher, John W.
;
Bush, Kimberly
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 December 2012 22(23):7201-7206
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7 . Academic Journal
Discovery of pyrazole carboxylic acids as potent inhibitors of rat long chain l-2-hydroxy acid oxidase
저자
by
Barawkar, Dinesh A.
;
Bandyopadhyay, Anish
;
Deshpande, Anil
;
Koul, Summon
;
Kandalkar, Sachin
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 July 2012 22(13):4341-4347
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7 . Academic Journal
MK-8825: A potent and selective CGRP receptor antagonist with good oral activity in rats
저자
by
Bell, Ian M.
;
Stump, Craig A.
;
Gallicchio, Steven N.
;
Staas, Donnette D.
;
Zartman, C. Blair
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 June 2012 22(12):3941-3945
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7 . Academic Journal
Discovery of pyrrolidine-based β-secretase inhibitors: Lead advancement through conformational design for maintenance of ligand binding efficiency
저자
by
Stachel, Shawn J.
;
Steele, Thomas G.
;
Petrocchi, Alessia
;
Haugabook, Sharie J.
;
McGaughey, Georgia
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 January 2012 22(1):240-244
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7 . Academic Journal
Identification of a novel RAMP-independent CGRP receptor antagonist
저자
by
Zartman, C. Blair
;
Bell, Ian M.
;
Gallicchio, Steven N.
;
Graham, Samuel L.
;
Kane, Stefanie A.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2011 21(22):6705-6708
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7 . Academic Journal
Orally bioavailable imidazoazepanes as calcitonin gene-related peptide (CGRP) receptor antagonists: Discovery of MK-2918
저자
by
Paone, Daniel V.
;
Nguyen, Diem N.
;
Shaw, Anthony W.
;
Burgey, Christopher S.
;
Potteiger, Craig M.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2011 21(9):2683-2686
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